SCHEMBL3819737

SCHEMBL3819737

CC1(C)CCC(c2ccc(Cl)cc2)=C(CN2CCN3c4ccc(C(=O)O)cc4CC[C@@H]3C2)C1

nearest known ligand 0.60

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
BCL2L1 Q07817 9/20 0.60
BCL2 P10415 10/20 0.49
DRD2 P14416 1/20 0.43
DRD4 P21917 1/20 0.43
CETP P11597 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5131603 0.99 BCL2L1 (0.59) BCL2L1BCL2DRD2DRD4CETP
SCHEMBL5128722 0.93 BCL2L1 (0.61) BCL2L1BCL2CETP
SCHEMBL5128718 0.93 BCL2L1 (0.61) BCL2L1BCL2CETP
Hydrochloric Acid SCHEMBL5129185 0.92 BCL2L1 (0.60) BCL2L1BCL2CETP
SCHEMBL30857750 0.86 BCL2L1 (0.58) BCL2L1BCL2CETP
SCHEMBL30857660 0.86 BCL2L1 (0.58) BCL2L1BCL2CETP
SCHEMBL3819200 0.85 DRD3 (0.40) BCL2L1DRD2DRD4
SCHEMBL4787539 0.85 DRD3 (0.40) BCL2L1DRD2DRD4
SCHEMBL30857714 0.84 BCL2L1 (0.57) BCL2L1BCL2CETP
Hydrochloric Acid SCHEMBL5129273 0.82 DRD2 (0.49) DRD2DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953161-B1 New tricyclic derivatives, method of preparing same and pharmaceutical compositions containing them SERVIER LAB (FR) 2009-08-26 EP disclosed
WO-2008110691-A1 NOVEL TRICYCLIC DERIVATIVES, METHOD FOR PREPARING SAME AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME LES LABORATOIRES SERVIER (FR) 2008-09-18 WO disclosed
US-20080188460-A1 Tricyclic compounds, a process for their preparation and pharmaceutical compositions containing them LES LABORATOIRES SERVIER (FR) 2008-08-07 US disclosed
EP-1953161-A1 New tricyclic derivatives, method of preparing same and pharmaceutical compositions containing them Les Laboratoires Servier (FR) 2008-08-06 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080188460-A1 Tricyclic compounds, a process for their preparation and pharmaceutical compositions containing them BAX, BCL2, CASP3 BCL2L1 45/4885BCL2 2/4885DRD2 2487/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.