SCHEMBL3824671

SCHEMBL3824671

NS(=O)(=O)c1ccc2c3c(ccc2c1)NCC3

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 7/20 0.52
CA2 P00918 7/20 0.52
CA12 O43570 4/20 0.52
CA9 Q16790 4/20 0.52
LMNA P02545 1/20 0.44
ADRA2A P08913 1/20 0.40
PNMT P11086 1/20 0.40
ADRA2B P18089 1/20 0.40
ADRA2C P18825 1/20 0.40
CA7 P43166 2/20 0.38
CA14 Q9ULX7 2/20 0.38
ALPL P05186 1/20 0.37
ALPI P09923 1/20 0.37
PKM P14618 1/20 0.37
PLG P00747 1/20 0.36
PLAU P00749 1/20 0.36
PLAT P00750 1/20 0.36
NOTUM Q6P988 1/20 0.36
ROCK1 Q13464 1/20 0.34
MAPT P10636 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29710882 0.74 CA1 (0.81) CA1CA2CA12CA9ADRA2A
SCHEMBL3238863 0.74 CA1 (0.81) CA1CA2CA12CA9ADRA2A
SCHEMBL30210907 0.72 CA2 (0.62) CA1CA2CA12CA9LMNA
SCHEMBL9770899 0.72 KDM4E (0.51) PLAUNOTUMMAPTCDK2
SCHEMBL4230983 0.71 CA1 (0.61) CA1CA2CA12CA9ADRA2A
SCHEMBL30664965 0.71 CA1 (0.61) CA1CA2CA12CA9ADRA2A
SCHEMBL5753987 0.70 ALDH1A1 (0.55) LMNAADRA2AADRA2BADRA2CMAPT
SCHEMBL31231831 0.69 CA1 (1.00) CA1CA2CA12CA9LMNA
SCHEMBL4162141 0.69 CA1 (1.00) CA1CA2CA12CA9LMNA
SCHEMBL9839080 0.69 LMNA (0.82) CA1CA2CA12CA9LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1809603-A4 NITROBENZINDOLES AND THEIR USE IN CANCER THERAPY AUCKLAND UNISERVICES LTD (NZ) 2009-09-02 EP claimed
EP-1809603-A1 NITROBENZINDOLES AND THEIR USE IN CANCER THERAPY Auckland Uniservices Limited (NZ) 2007-07-25 EP claimed
WO-2006043839-A1 NITROBENZINDOLES AND THEIR USE IN CANCER THERAPY AUCKLAND UNISERVICES LIMITED (NZ) 2006-04-27 WO claimed