SCHEMBL3825571

SCHEMBL3825571

CC(C)C(=O)N1CCC(Nc2ccc(C#N)c(Cl)c2)C1

nearest known ligand 0.49

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PGR P06401 10/20 0.49
CYP2C9 P11712 10/20 0.49
CYP2D6 P10635 8/20 0.49
DPP4 P27487 3/20 0.47
KCNH2 Q12809 1/20 0.47
HDAC8 Q9BY41 1/20 0.46
HDAC6 Q9UBN7 1/20 0.46
AR P10275 1/20 0.41
SPR P35270 1/20 0.41
EPHX2 P34913 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3825564 1.00 PGR (0.49) PGRCYP2C9CYP2D6DPP4KCNH2
SCHEMBL3025009 0.86 DPP4 (0.50) PGRCYP2C9CYP2D6DPP4HDAC8
SCHEMBL13238912 0.82 ALDH1A1 (0.53) PGRCYP2C9CYP2D6DPP4HDAC8
SCHEMBL3024142 0.79 PGR (0.51) PGRCYP2C9CYP2D6DPP4KCNH2
SCHEMBL380969 0.77 ALDH1A1 (0.61) DPP4HDAC8HDAC6L3MBTL1
SCHEMBL3037282 0.76 PGR (0.51) PGRCYP2C9CYP2D6DPP4KCNH2
SCHEMBL3326284 0.76 DPP4 (0.49) PGRDPP4KCNH2HDAC8HDAC6
SCHEMBL3326291 0.76 DPP4 (0.49) PGRDPP4KCNH2HDAC8HDAC6
SCHEMBL3326316 0.76 DPP4 (0.49) PGRDPP4KCNH2HDAC8HDAC6
SCHEMBL12043205 0.75 AR (0.44) PGRCYP2C9CYP2D6DPP4KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2094269-A1 PYRROLIDINANILINES Smithkline Beecham Corporation (US) 2009-09-02 EP disclosed
WO-2008077089-A1 PYRROLIDINANILINES SMITHKLINE BEECHAM CORPORATION (US) 2008-06-26 WO disclosed