SCHEMBL3825653

SCHEMBL3825653

Fc1ccccc1ON1CCCCC1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.46
KDM4E B2RXH2 4/20 0.46
KMT2A Q03164 4/20 0.46
MEN1 O00255 3/20 0.46
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2D6 P10635 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
PKM P14618 1/20 0.39
HPGD P15428 2/20 0.37
TSHR P16473 1/20 0.37
MAPK1 P28482 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
FKBP1A P62942 1/20 0.36
HTT P42858 1/20 0.36
GAA P10253 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23850504 0.98 ALDH1A1 (0.47) ALDH1A1KDM4EKMT2AMEN1CYP1A2
SCHEMBL23850464 0.94 ALDH1A1 (0.44) ALDH1A1KDM4EKMT2AMEN1CYP1A2
SCHEMBL3073484 0.82 KDM4E (0.47) ALDH1A1KDM4ETSHRSMN1; SMN2HTT
Trifluoroacetic Acid SCHEMBL23853666 0.80 CXCL8 (0.41) ALDH1A1KDM4EKMT2AMEN1CYP1A2
SCHEMBL22817829 0.78 SLC6A2 (0.43) ALDH1A1KDM4EKMT2AMEN1CYP1A2
SCHEMBL3129171 0.78 ALDH1A1 (0.40) ALDH1A1KDM4EKMT2AMEN1CYP1A2
SCHEMBL19039738 0.77 TRPC3 (0.35) ALDH1A1KDM4EKMT2AMEN1CYP1A2
SCHEMBL11548078 0.76 CA12 (0.52) ALDH1A1KMT2AMEN1PKMTSHR
SCHEMBL4504681 0.76 ALDH1A1 (0.44) ALDH1A1KDM4EKMT2AHPGDTSHR
SCHEMBL10701429 0.76 KEAP1 (0.47) ALDH1A1KDM4ECYP1A2CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2099755-A2 ACETYLENE DERIVATIVES AS STEAROYL COA DESATURASE INHIBITORS Glenmark Pharmaceuticals S.A. (CH) 2009-09-16 EP claimed
WO-2008062276-A2 ACETYLENE DERIVATIVES AS STEAROYL COA DESATURASE INHIBITORS GLENMARK PHARMACEUTICALS S.A. (US) 2008-05-29 WO claimed
CN-115210225-A Substituted aminoquinolones as immuno-activated DGKALPHA inhibitors 拜耳公司 2022-10-18 CN disclosed