SCHEMBL3826

SCHEMBL3826

C[C@]12C=CC(=O)C=C1CC[C@@H]1[C@@H]2[C@@H](O)C[C@@]2(C)[C@H]1CC[C@]2(O)C(=O)OCCl

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PGR P06401 5/20 0.76
HIF1A Q16665 5/20 0.76
NR3C1 P04150 13/20 0.74
HSD17B10 Q99714 2/20 0.74
ABCB11 O95342 2/20 0.74
CYP3A4 P08684 2/20 0.74
TNF P01375 1/20 0.74
IL6 P05231 1/20 0.74
SERPINA6 P08185 1/20 0.74
NR3C2 P08235 1/20 0.74
AR P10275 1/20 0.74
GLUL P15104 1/20 0.74
ADAM17 P78536 1/20 0.74
GPBAR1 Q8TDU6 1/20 0.74
CYP2C19 P33261 1/20 0.74
ABCC3 O15438 1/20 0.72
NR1I2 O75469 1/20 0.72
LMNA P02545 3/20 0.66
USP2 O75604 1/20 0.57
CYP2D6 P10635 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23974880 1.00 PGR (0.76) PGRHIF1ANR3C1HSD17B10ABCB11
SCHEMBL1685716 0.92 PGR (0.77) PGRHIF1ANR3C1HSD17B10ABCB11
SCHEMBL5098424 0.92 PGR (0.77) PGRHIF1ANR3C1HSD17B10ABCB11
SCHEMBL12969465 0.89 NR3C1 (0.76) PGRHIF1ANR3C1HSD17B10ABCB11
SCHEMBL12738238 0.89 NR3C1 (0.76) PGRHIF1ANR3C1HSD17B10ABCB11
SCHEMBL1685803 0.89 NR3C1 (0.76) PGRHIF1ANR3C1HSD17B10ABCB11
SCHEMBL13379819 0.89 NR3C1 (0.76) PGRHIF1ANR3C1HSD17B10ABCB11
SCHEMBL15796471 0.89 NR3C1 (0.76) PGRHIF1ANR3C1HSD17B10ABCB11
SCHEMBL5098329 0.89 NR3C1 (0.76) PGRHIF1ANR3C1HSD17B10ABCB11
SCHEMBL11856593 0.88 NR3C1 (0.84) PGRHIF1ANR3C1HSD17B10ABCB11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 8117 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260137657-A1 METHODS AND COMPOSITIONS FOR TREATING GLUCOCORTICOID EXCESS SPARROW PHARMACEUTICALS INC (US) 2026-05-21 US claimed
US-20260137558-A1 OPHTHALMIC DEVICE Able Tx Ltd. (IL) 2026-05-21 US claimed
US-20260137656-A1 METHODS AND COMPOSITIONS FOR TREATING GLUCOCORTICOID EXCESS SPARROW PHARMACEUTICALS INC (US) 2026-05-21 US claimed
WO-2026100654-A1 NUCLEIC ACID INTRODUCTION AID, NUCLEIC ACID INTRODUCTION AGENT, AND NUCLEIC ACID INTRODUCTION METHOD 株式会社インファーマシア 2026-05-15 WO claimed
US-12616654-B2 Stainless steel can for pressurised metered dose inhalers CHIESI FARMACEUTICI S.P.A. (IT) 2026-05-05 US claimed
US-20260108610-A1 Drug-Resistant Immune Cells and Methods of Use Thereof REGENTS OF THE UNIVERSITY OF MINNESOTA 2026-04-23 US claimed
EP-4724079-A2 METHODS AND COMPOSITIONS FOR THE TREATMENT OF AGE-RELATED MACULAR DEGENERATION Stealth BioTherapeutics Inc. (US) 2026-04-15 EP claimed
US-12599556-B2 Ophthalmic compositions BIOTHERAVISION INC. (US) 2026-04-14 US claimed
US-20260091017-A1 TREATMENTS FOR INFLAMMATION AUCKLAND UNISERVICES LTD (NZ) 2026-04-02 US claimed
EP-4259102-B1 COMPOSITIONS AND METHODS FOR MUCOSAL DRUG DELIVERY UNIV CALIFORNIA (US) 2026-03-11 EP claimed
CN-1315852-A Medicinal aerosol formulations JAGO RES AG (CH) 2001-10-03 CN claimed
EP-1131059-A1 DRY POWDER FOR INHALATION JAGO RESEARCH AG (CH) 2001-09-12 EP claimed
WO-2001058438-A1 OPHTHALMIC USE OF ALPHA ADRENERGIC BLOCKING AGENTS GALIN MILES A (US) 2001-08-16 WO claimed
EP-1102579-A1 MEDICINAL AEROSOL FORMULATIONS JAGO RESEARCH AG (CH) 2001-05-30 EP claimed
WO-2001022955-A2 NOVEL COMBINATION OF LOTEPREDNOL AND ANTIHISTAMINES VIATRIS GMBH & CO. KG (DE) 2001-04-05 WO claimed
US-6106819-A Methods of treating headache and functional extraocular and intraocular myotendinitis SUCHER DAVID F (US) 2000-08-22 US claimed
EP-1014943-A1 MEDICAL AEROSOL FORMULATIONS Jago Research AG (CH) 2000-07-05 EP claimed
WO-2000028979-A1 DRY POWDER FOR INHALATION JAGO RESEARCH AG (CH) 2000-05-25 WO claimed
WO-2000007567-A1 MEDICINAL AEROSOL FORMULATIONS JAGO RESEARCH AG (CH) 2000-02-17 WO claimed
WO-1998034595-A1 MEDICAL AEROSOL FORMULATIONS JAGO RESEARCH AG (CH) 1998-08-13 WO claimed