SCHEMBL3827366

SCHEMBL3827366

CC(C)(C)OC(=O)N(Br)c1ccc2ccc(S(C)(=O)=O)cc2c1

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 2/20 0.37
AKR1C2 P52895 2/20 0.37
GPR119 Q8TDV5 5/20 0.35
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
POLB P06746 1/20 0.34
ACACB O00763 1/20 0.34
TMEM97 Q5BJF2 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
KAT6A Q92794 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
NQO2 P16083 1/20 0.33
MTNR1A P48039 1/20 0.33
MTNR1B P49286 1/20 0.33
GAA P10253 1/20 0.33
NR1H2 P55055 1/20 0.32
NR1H3 Q13133 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1007952 0.83 GPR119 (0.42) GPR119NR1H2NR1H3
SCHEMBL7714859 0.82 ALDH1A1 (0.40) MEN1KMT2APOLBSMN1; SMN2
SCHEMBL3831845 0.80 CNR2 (0.53) MEN1KMT2A
SCHEMBL3827000 0.79 CYP2A6 (0.45) GPR119MEN1KMT2ANPC1RAB9A
SCHEMBL3566610 0.78 AKR1C3 (0.33) AKR1C3AKR1C2GPR119TMEM97KAT6A
SCHEMBL3825115 0.77 NCEH1 (0.42) GPR119
SCHEMBL3827550 0.76 AKR1C3 (0.50) AKR1C3AKR1C2MEN1KMT2APOLB
SCHEMBL7715157 0.75 CA12 (0.45) NPC1RAB9A
SCHEMBL3559616 0.74 AKR1C3 (0.36) AKR1C3AKR1C2GPR119ACACBTMEM97
SCHEMBL3554857 0.72 KAT6A (0.55) ACACBKAT6A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1809603-A4 NITROBENZINDOLES AND THEIR USE IN CANCER THERAPY AUCKLAND UNISERVICES LTD (NZ) 2009-09-02 EP disclosed
EP-1809603-A1 NITROBENZINDOLES AND THEIR USE IN CANCER THERAPY Auckland Uniservices Limited (NZ) 2007-07-25 EP disclosed
WO-2006043839-A1 NITROBENZINDOLES AND THEIR USE IN CANCER THERAPY AUCKLAND UNISERVICES LIMITED (NZ) 2006-04-27 WO disclosed