SCHEMBL7714859

SCHEMBL7714859

CC(C)(C)OC(=O)N(Br)c1ccc2ccc(OS(C)(=O)=O)cc2c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.40
MEN1 O00255 3/20 0.35
KMT2A Q03164 3/20 0.35
ESR1 P03372 1/20 0.35
ATM Q13315 1/20 0.35
ESR2 Q92731 1/20 0.35
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA9 Q16790 1/20 0.33
SMN1; SMN2 Q16637 2/20 0.32
NCEH1 Q6PIU2 1/20 0.32
LMNA P02545 3/20 0.32
L3MBTL1 Q9Y468 2/20 0.32
PPARG P37231 1/20 0.32
HTT P42858 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
POLB P06746 1/20 0.31
KDM4E B2RXH2 1/20 0.31
MT-CO2 P00403 1/20 0.31
KEAP1 Q14145 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3827366 0.82 AKR1C3 (0.37) MEN1KMT2ASMN1; SMN2POLB
SCHEMBL7715157 0.81 CA12 (0.45) ALDH1A1CA1CA9NCEH1LMNA
SCHEMBL7718988 0.78 ALDH1A1 (0.38) ALDH1A1CA1CA2CA9SMN1; SMN2
SCHEMBL3827000 0.77 CYP2A6 (0.45) ALDH1A1MEN1KMT2AESR1ESR2
SCHEMBL3825115 0.75 NCEH1 (0.42) NCEH1PTPN1
SCHEMBL1007952 0.70 GPR119 (0.42)
SCHEMBL1007329 0.68 MT-CO2 (0.51) ALDH1A1MEN1KMT2ASMN1; SMN2TDP1
SCHEMBL1008034 0.68 MT-CO2 (0.39) ALDH1A1MEN1KMT2AATMSMN1; SMN2
SCHEMBL20364928 0.67 L3MBTL1 (0.56) ALDH1A1MEN1KMT2ACA1CA2
SCHEMBL4556628 0.67 ALOX15 (0.40) ALDH1A1MEN1KMT2AATMSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1214326-A1 INHIBITORS OF PRENYL-PROTEIN TRANSFERASE Merck & Co., Inc. (US) 2002-06-19 EP disclosed
WO-2001018006-A1 INHIBITORS OF PRENYL-PROTEIN TRANSFERASE MERCK & CO., INC. (US) 2001-03-15 WO disclosed