SCHEMBL3828429

SCHEMBL3828429

CNC(=O)c1sc2ccccc2c1N

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.67
HPGD P15428 4/20 0.67
MAPT P10636 3/20 0.67
KDM4E B2RXH2 3/20 0.67
MEN1 O00255 2/20 0.67
KMT2A Q03164 2/20 0.67
GLA P06280 2/20 0.67
GAA P10253 2/20 0.67
HSD17B10 Q99714 2/20 0.67
ALOX15 P16050 1/20 0.67
ATM Q13315 1/20 0.67
LIMK1 P53667 2/20 0.65
IKBKB O14920 2/20 0.65
GABRA1 P14867 1/20 0.54
GABRA5 P31644 1/20 0.54
HDAC1 Q13547 1/20 0.51
HDAC8 Q9BY41 1/20 0.51
HDAC6 Q9UBN7 1/20 0.51
OGG1 O15527 1/20 0.50
MAPK1 P28482 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29285354 0.85 OGG1 (0.69) ALDH1A1HPGDMAPTKDM4EMEN1
SCHEMBL15766514 0.81 LIMK1 (0.71) ALDH1A1HPGDMAPTKDM4EMEN1
SCHEMBL30173777 0.80 KDM4E (1.00) ALDH1A1HPGDMAPTKDM4EMEN1
SCHEMBL7984062 0.80 HDAC1 (0.79) ALDH1A1HPGDMAPTKDM4EMEN1
SCHEMBL1101766 0.80 KDM4E (1.00) ALDH1A1HPGDMAPTKDM4EMEN1
SCHEMBL1919937 0.79 LIMK1 (0.73) ALDH1A1HPGDMAPTKDM4EMEN1
SCHEMBL6609258 0.79 LIMK1 (1.00) ALDH1A1HPGDMAPTKDM4EMEN1
SCHEMBL4724459 0.78 KDM4E (0.70) ALDH1A1HPGDMAPTKDM4EMEN1
SCHEMBL11683541 0.75 ALDH1A1 (0.61) ALDH1A1HPGDMAPTKDM4EMEN1
SCHEMBL16581218 0.75 GABRA1 (0.77) ALDH1A1HPGDMAPTKDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1874295-A4 BENZOTHIOPHENE DERIVATIVES MERCK & CO INC (US) 2009-08-12 EP disclosed
EP-1874295-A1 BENZOTHIOPHENE DERIVATIVES Merck & Co., Inc. (US) 2008-01-09 EP disclosed
WO-2006115845-A1 BENZOTHIOPHENE DERIVATIVES MERCK & CO., INC. (US) 2006-11-02 WO disclosed