SCHEMBL3829336

SCHEMBL3829336

O=C(O)c1cnc2cncnc2n1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX15 P16050 3/20 0.50
ALDH1A1 P00352 2/20 0.50
HPGD P15428 1/20 0.50
HSD17B10 Q99714 1/20 0.50
AKR1B1 P15121 1/20 0.41
KDM4E B2RXH2 5/20 0.38
HCAR2 Q8TDS4 2/20 0.38
NAPRT Q6XQN6 2/20 0.38
PIK3CG P48736 1/20 0.36
LMNA P02545 2/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
TSHR P16473 2/20 0.33
P4HTM Q9NXG6 2/20 0.33
ACMSD Q8TDX5 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
P4HA1 P13674 1/20 0.33
MIF P14174 1/20 0.33
DPP4 P27487 1/20 0.33
DPP7 Q9UHL4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6317502 0.85 ALOX15 (0.50) ALOX15ALDH1A1HPGDHSD17B10AKR1B1
SCHEMBL28822491 0.81 PIK3CG (0.34) ALOX15ALDH1A1HPGDHSD17B10PIK3CG
SCHEMBL5564401 0.74 KDM4E (0.56) ALOX15ALDH1A1HPGDHSD17B10KDM4E
SCHEMBL316631 0.72 PIK3CG (0.44) PIK3CGEGFR
SCHEMBL316630 0.72 PIK3CG (0.37) PIK3CGEGFR
SCHEMBL9903399 0.71 ALDH1A1 (0.47) ALOX15ALDH1A1HPGDHSD17B10AKR1B1
Purine SCHEMBL10946421 0.71 ALDH1A1 (0.61) ALOX15ALDH1A1HPGDHSD17B10KDM4E
SCHEMBL6260367 0.70 ALOX15 (0.50) ALOX15ALDH1A1HPGDHSD17B10KDM4E
SCHEMBL11769997 0.70 ALDH1A1 (0.65) ALOX15ALDH1A1HPGDHSD17B10KDM4E
SCHEMBL3292267 0.70 PIK3CG (0.47) ALDH1A1HSD17B10PIK3CGTSHREGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2102210-A2 COMPOUNDS USEFUL AS PROTEIN KINASE INHIBITORS Vertex Pharmceuticals Incorporated (US) 2009-09-23 EP disclosed
WO-2008076392-A2 COMPOUNDS USEFUL AS PROTEIN KINASE INHIBITORS VERTEX PHARMACEUTICALS INCORPORATED (US) 2008-06-26 WO disclosed