SCHEMBL3836027

SCHEMBL3836027

N#Cc1cc(C#N)cc(Oc2cc(CC(=O)Nc3ccc(OCC(=O)O)cc3)ccc2Cl)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RORC P51449 1/20 0.43
MAPT P10636 3/20 0.42
MAPK1 P28482 1/20 0.42
HTT P42858 2/20 0.41
AKR1B1 P15121 1/20 0.41
KMT2A Q03164 3/20 0.41
GAA P10253 2/20 0.41
CSF1R P07333 1/20 0.41
RET P07949 1/20 0.41
PDGFRB P09619 1/20 0.41
KIT P10721 1/20 0.41
PDGFRA P16234 1/20 0.41
DDR1 Q08345 1/20 0.41
MEN1 O00255 2/20 0.41
ALDH1A1 P00352 1/20 0.41
NPC1 O15118 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
HPGD P15428 1/20 0.40
RAB9A P51151 1/20 0.40
LMNA P02545 3/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3837011 0.91 NR1H4 (0.49) RORCMAPTHTTKMT2AGAA
SCHEMBL2639293 0.90 RORC (0.44) RORCMAPTHTTKMT2AGAA
SCHEMBL2639768 0.90 MAPT (0.47) RORCMAPTMAPK1HTTKMT2A
SCHEMBL2638287 0.89 RORC (0.44) RORCMAPTMAPK1HTTKMT2A
SCHEMBL2638078 0.89 LMNA (0.51) RORCMAPTKMT2AMEN1ALDH1A1
SCHEMBL3218393 0.88 RORC (0.43) RORCMAPTHTTKMT2AGAA
SCHEMBL3835920 0.88 RORC (0.45) RORCMAPTHTTKMT2AGAA
SCHEMBL2640022 0.88 RORC (0.46) RORCMAPTHTTKMT2AGAA
SCHEMBL3836762 0.87 RORC (0.42) RORCMAPTHTTKMT2AGAA
SCHEMBL3835196 0.86 MAPT (0.43) RORCMAPTMAPK1HTTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1742908-B1 NON-NUCLEOSIDE REVERSE TRANSCRIPTASE INHIBITORS HOFFMANN LA ROCHE (CH) 2009-11-11 EP claimed