SCHEMBL3836268

SCHEMBL3836268

Nc1nc2c(c(=O)[nH]1)NCN2CCCO

nearest known ligand 0.61

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HPRT1 P00492 9/20 0.61
TK1 P04183 1/20 0.40
NOS1 P29475 4/20 0.35
CYP1A2 P05177 1/20 0.34
PNP P00491 1/20 0.33
NOS3 P29474 1/20 0.33
NOS2 P35228 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL571646 0.96 HPRT1 (0.60) HPRT1TK1NOS1CYP1A2PNP
SCHEMBL3793007 0.86 HPRT1 (0.58) HPRT1TK1NOS1CYP1A2PNP
SCHEMBL9739844 0.85 HPRT1 (0.60) HPRT1NOS1PNPNOS3NOS2
SCHEMBL10511442 0.85 HPRT1 (0.53) HPRT1TK1NOS1CYP1A2
SCHEMBL9663134 0.85 HPRT1 (0.55) HPRT1TK1NOS1
SCHEMBL6061495 0.84 HPRT1 (0.58) HPRT1TK1NOS1CYP1A2PNP
SCHEMBL489058 0.84 HPRT1 (0.56) HPRT1NOS1PNPNOS3NOS2
SCHEMBL9662657 0.84 HPRT1 (0.56) HPRT1NOS1CYP1A2NOS3NOS2
SCHEMBL8842510 0.83 HPRT1 (0.58) HPRT1NOS1PNP
SCHEMBL9364441 0.83 HPRT1 (0.60) HPRT1NOS1PNPNOS3NOS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 21 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0143987-B1 THERAPEUTIC COMPOSITIONS ENDOWED WITH ANTIVIRAL ACTIVITY Stendardi, Anna Gioia (IT) 1989-02-22 EP claimed
US-7590493-B2 Methods for determining hepatotoxins OCIMUM BIOSOLUTIONS, INC. (US) 2009-09-15 US disclosed
US-20090220970-A1 MOLECULAR TOXICOLOGY MODELING OCIMUM BIOSOLUTIONS, INC. 2009-09-03 US disclosed
US-7426441-B2 Methods for determining renal toxins OCIMUM BIOSOLUTIONS, INC. (US) 2008-09-16 US disclosed
US-7415358-B2 Molecular toxicology modeling OCIMUM BIOSOLUTIONS, INC. (US) 2008-08-19 US disclosed
EP-1476747-A4 MOLECULAR HEPATOTOXICOLOGY MODELING OCIMUM BIOSOLUTIONS INC (US) 2008-06-11 EP disclosed
US-20070124086-A1 Molecular nephrotoxicology modeling OCIMUM BIOSOLUTIONS, INC. 2007-05-31 US disclosed
US-20070093969-A1 Molecular nephrotoxicology modeling OCIMUM BIOSOLUTIONS, INC. 2007-04-26 US disclosed
US-20070043515-A1 Molecular toxicology modeling GENE LOGIC, INC. 2007-02-22 US disclosed
US-20070027634-A1 Molecular hepatotoxicology modeling OCIMUM BIOSOLUTIONS, INC. 2007-02-01 US disclosed
EP-1392871-A4 MOLECULAR TOXICOLOGY MODELING GENE LOGIC INC (US) 2006-04-19 EP disclosed
US-20060078900-A1 Molecular toxicology modeling GENE LOGIC, INC. 2006-04-13 US disclosed
EP-1563295-A2 MOLECULAR NEPHROTOXICOLOGY MODELING Gene Logic, Inc. (US) 2005-08-17 EP disclosed
EP-1476747-A2 MOLECULAR HEPATOTOXICOLOGY MODELING Gene Logic, Inc. (US) 2004-11-17 EP disclosed
WO-2004048598-A2 MOLECULAR NEPHROTOXICOLOGY MODELING GENE LOGIC, INC. (US) 2004-06-10 WO disclosed
US-20040072160-A1 Molecular toxicology modeling OCIMUM BIOSOLUTIONS, INC. 2004-04-15 US disclosed
EP-1392871-A2 MOLECULAR TOXICOLOGY MODELING Gene Logic, Inc. (US) 2004-03-03 EP disclosed
WO-2003064624-A2 MOLECULAR HEPATOTOXICOLOGY MODELING GENE LOGIC, INC. (US) 2003-08-07 WO disclosed
WO-2002095000-A2 MOLECULAR TOXICOLOGY MODELING GENE LOGIC, INC. (US) 2002-11-28 WO disclosed
CN-1058598-A NEW LINKER FOR BIOACTIVE AGENTS ERBA CARLO SPA (IT) 1992-02-12 CN disclosed