SCHEMBL3836451

SCHEMBL3836451

CCOC(=O)C(CC(=O)CC)=NC

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.40
NPSR1 Q6W5P4 3/20 0.39
GLO1 Q04760 1/20 0.39
ALDH1A1 P00352 5/20 0.39
CYP2D6 P10635 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
MGAM O43451 1/20 0.38
GAA P10253 1/20 0.38
SI P14410 1/20 0.38
MGAM2 Q2M2H8 1/20 0.38
SOAT1 P35610 1/20 0.38
MEN1 O00255 4/20 0.38
KMT2A Q03164 4/20 0.38
EGLN1 Q9GZT9 1/20 0.37
APOBEC3A P31941 1/20 0.36
APOBEC3G Q9HC16 1/20 0.36
LMNA P02545 3/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5706998 0.83 NPSR1 (0.45) MAPTNPSR1GLO1ALDH1A1CYP2D6
SCHEMBL5706996 0.83 NPSR1 (0.45) MAPTNPSR1GLO1ALDH1A1CYP2D6
SCHEMBL20778292 0.81 MAPT (0.38) MAPTNPSR1GLO1ALDH1A1CYP2D6
SCHEMBL29134126 0.81 MAPT (0.38) MAPTNPSR1GLO1ALDH1A1CYP2D6
SCHEMBL19168953 0.75 ALDH1A1 (0.48) MAPTNPSR1GLO1ALDH1A1CYP2D6
SCHEMBL7240646 0.74 TDP1 (0.41) TDP1
SCHEMBL1178944 0.74 MGAM (0.44) MAPTNPSR1GLO1ALDH1A1CYP2D6
SCHEMBL28622235 0.70 APOBEC3A (0.51) MAPTNPSR1GLO1ALDH1A1CYP2D6
SCHEMBL26325159 0.70 APOBEC3A (0.51) MAPTNPSR1GLO1ALDH1A1CYP2D6
SCHEMBL18590176 0.69 MAPT (0.46) MAPTNPSR1GLO1ALDH1A1CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0946508-B1 NITROGEN CONTAINING HETEROAROMATICS AS FACTOR Xa INHIBITORS BRISTOL MYERS SQUIBB PHARMA CO (US) 2009-09-23 EP disclosed
US-6020357-A CARDIOVASCULAR DISORDERS; ANTCOAGULANTS DUPONT PHARMACEUTICALS COMPANY (US) 2000-02-01 US disclosed