SCHEMBL3836764

SCHEMBL3836764

CC(O)(Cc1cc(F)cc(F)c1)CC1CN(C(c2ccc(Cl)cc2)c2cccc(C#N)c2)C1

nearest known ligand 0.40

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 15/20 0.40
CNR2 P34972 11/20 0.40
MGLL Q99685 3/20 0.37
MEN1 O00255 1/20 0.36
GLA P06280 1/20 0.36
TSHR P16473 1/20 0.36
KMT2A Q03164 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
ALDH1A1 P00352 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1569103 0.91 CNR1 (0.41) CNR1CNR2MGLLMEN1GLA
SCHEMBL4080122 0.90 CNR1 (0.40) CNR1CNR2MGLLMEN1GLA
SCHEMBL5727699 0.87 CNR1 (0.38) CNR1CNR2MGLLMEN1GLA
SCHEMBL4787427 0.85 CNR1 (0.36) CNR1CNR2MGLLMEN1GLA
SCHEMBL4683968 0.84 CNR1 (0.37) CNR1CNR2MGLLMEN1GLA
SCHEMBL5727680 0.84 MGLL (0.41) CNR1CNR2MGLLMEN1GLA
SCHEMBL5727485 0.82 TSHR (0.37) CNR1CNR2MGLLMEN1GLA
SCHEMBL4968374 0.82 CNR1 (0.39) CNR1CNR2MGLL
SCHEMBL4681476 0.81 CNR1 (0.34) CNR1CNR2MGLLMEN1GLA
SCHEMBL5727631 0.81 MEN1 (0.37) CNR1CNR2MGLLMEN1GLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1636181-A1 SUBSTITUTED 3-ALKYL AND 3-ALKENYL AZETIDINE DERIVATIVES Merck & Co., Inc. (US) 2006-03-22 EP claimed
WO-2005000809-A1 SUBSTITUTED 3-ALKYL AND 3-ALKENYL AZETIDINE DERIVATIVES MERCK & CO., INC. (US) 2005-01-06 WO claimed
EP-2120569-A2 SPIROCHROMANON DERIVATIVES Merck & Co., Inc. (US) 2009-11-25 EP disclosed
EP-2111406-A1 SUBSTITUTED SPIROCHROMANONE DERIVATIVES AS ACC INHIBITORS Merck & Co., Inc. (US) 2009-10-28 EP disclosed
WO-2008088688-A1 SUBSTITUTED SPIROCHROMANONE DERIVATIVES AS ACC INHIBITORS MERCK & CO., INC. (US) 2008-07-24 WO disclosed
WO-2008088692-A2 SPIROCHROMANON DERIVATIVES MERCK & CO., INC. (US) 2008-07-24 WO disclosed
EP-1636181-A1 SUBSTITUTED 3-ALKYL AND 3-ALKENYL AZETIDINE DERIVATIVES Merck & Co., Inc. (US) 2006-03-22 EP disclosed
WO-2005000809-A1 SUBSTITUTED 3-ALKYL AND 3-ALKENYL AZETIDINE DERIVATIVES MERCK & CO., INC. (US) 2005-01-06 WO disclosed