SCHEMBL4683968

SCHEMBL4683968

CC(F)(Cc1cc(F)cc(C(=O)O)c1)CC1CN(C(c2ccc(Cl)cc2)c2cccc(C#N)c2)C1

nearest known ligand 0.37

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 15/20 0.37
CNR2 P34972 11/20 0.37
MGLL Q99685 3/20 0.37
MEN1 O00255 1/20 0.34
GLA P06280 1/20 0.34
TSHR P16473 1/20 0.34
KMT2A Q03164 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
KLKB1 P03952 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
KCNH2 Q12809 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4968374 0.92 CNR1 (0.39) CNR1CNR2MGLLKLKB1CYP3A4
SCHEMBL4080122 0.91 CNR1 (0.40) CNR1CNR2MGLLMEN1GLA
SCHEMBL4684089 0.90 MGLL (0.36) CNR1CNR2MGLLKLKB1CYP2D6
SCHEMBL5727699 0.90 CNR1 (0.38) CNR1CNR2MGLLMEN1GLA
SCHEMBL4787427 0.87 CNR1 (0.36) CNR1CNR2MGLLMEN1GLA
SCHEMBL5727680 0.85 MGLL (0.41) CNR1CNR2MGLLMEN1GLA
SCHEMBL4681878 0.85 SLC6A9 (0.37) MEN1TSHRKMT2ACYP3A4CYP2D6
SCHEMBL4681581 0.85 ELANE (0.38) MGLLMEN1GLATSHRKMT2A
SCHEMBL4966303 0.84 MGLL (0.40) MGLLMEN1GLATSHRKMT2A
SCHEMBL4681476 0.84 CNR1 (0.34) CNR1CNR2MGLLMEN1GLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1960392-A2 HETEROCYCLE-SUBSTITUTED 3-ALKYL AZETIDINE DERIVATIVES Merck & Co., Inc. (US) 2008-08-27 EP disclosed
EP-1954692-A1 HETEROCYCLE-SUBSTITUTED 3-ALKYL AZETIDINE DERIVATIVES Merck and Co., Inc. (US) 2008-08-13 EP disclosed
WO-2007064566-A2 HETEROCYCLE-SUBSTITUTED 3-ALKYL AZETIDINE DERIVATIVES MERCK & CO., INC. (US) 2007-06-07 WO disclosed
WO-2007062193-A1 HETEROCYCLE-SUBSTITUTED 3-ALKYL AZETIDINE DERIVATIVES MERCK & CO., INC. (US) 2007-05-31 WO disclosed