SCHEMBL5727680

SCHEMBL5727680

CC(F)(Cc1cc(F)cc(F)c1)CC1CN(C(c2ccc(F)cc2)c2cccc(C#N)c2)C1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MGLL Q99685 2/20 0.41
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
TSHR P16473 2/20 0.38
NPSR1 Q6W5P4 2/20 0.38
GLA P06280 1/20 0.38
ALDH1A1 P00352 2/20 0.36
POLB P06746 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.33
CNR1 P21554 1/20 0.33
CNR2 P34972 1/20 0.33
NR3C1 P04150 1/20 0.33
NR3C2 P08235 1/20 0.33
ACHE P22303 1/20 0.32
FADS1 O60427 2/20 0.32
KDM4D Q6B0I6 1/20 0.32
DGKA P23743 1/20 0.32
DGKZ Q13574 1/20 0.32
GAA P10253 1/20 0.32
HSD17B10 Q99714 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5727485 0.94 TSHR (0.37) MGLLMEN1KMT2ATSHRNPSR1
SCHEMBL4080122 0.94 CNR1 (0.40) MGLLMEN1KMT2ATSHRNPSR1
SCHEMBL5727631 0.94 MEN1 (0.37) MGLLMEN1KMT2ATSHRNPSR1
SCHEMBL4072255 0.93 MEN1 (0.37) MGLLMEN1KMT2ATSHRNPSR1
SCHEMBL5727699 0.90 CNR1 (0.38) MGLLMEN1KMT2ATSHRNPSR1
SCHEMBL4684882 0.90 MEN1 (0.36) MGLLMEN1KMT2ATSHRNPSR1
SCHEMBL4966303 0.88 MGLL (0.40) MGLLMEN1KMT2ATSHRNPSR1
SCHEMBL4787427 0.88 CNR1 (0.36) MGLLMEN1KMT2ATSHRNPSR1
SCHEMBL5727486 0.86 MGLL (0.37) MGLLMEN1KMT2ATSHRNPSR1
SCHEMBL1569103 0.85 CNR1 (0.41) MGLLMEN1KMT2ATSHRNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1636181-A1 SUBSTITUTED 3-ALKYL AND 3-ALKENYL AZETIDINE DERIVATIVES Merck & Co., Inc. (US) 2006-03-22 EP claimed
WO-2005000809-A1 SUBSTITUTED 3-ALKYL AND 3-ALKENYL AZETIDINE DERIVATIVES MERCK & CO., INC. (US) 2005-01-06 WO claimed