SCHEMBL3838003

SCHEMBL3838003

COc1ccc(C(=O)CN2CCN(CC(O)c3ccccc3)CC2)cc1

nearest known ligand 0.61

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.61
LMNA P02545 5/20 0.61
KDM4E B2RXH2 2/20 0.61
MITF O75030 2/20 0.57
SMN1; SMN2 Q16637 2/20 0.57
HIF1A Q16665 1/20 0.57
KMT2A Q03164 3/20 0.55
MEN1 O00255 2/20 0.54
TP53 P04637 1/20 0.54
KDR P35968 1/20 0.53
GAA P10253 1/20 0.53
MAPT P10636 3/20 0.53
HTT P42858 1/20 0.53
CHRM3 P20309 1/20 0.52
SLC6A4 P31645 1/20 0.51
SLC6A3 Q01959 1/20 0.51
HTR1A P08908 1/20 0.51
IGF1R P08069 1/20 0.51
NPSR1 Q6W5P4 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4875943 0.99 ALDH1A1 (0.60) ALDH1A1LMNAKDM4EMITFSMN1; SMN2
SCHEMBL3837620 0.88 HTR1A (0.67) ALDH1A1LMNAKDM4EKMT2AMEN1
Hydrochloric Acid SCHEMBL4811673 0.87 HTR1A (0.66) ALDH1A1LMNAKDM4EKMT2AMEN1
SCHEMBL3838547 0.87 SLC6A4 (0.60) ALDH1A1KDM4EKMT2AMEN1GAA
Hydrochloric Acid SCHEMBL3840088 0.86 SLC6A4 (0.59) ALDH1A1KDM4EMITFSMN1; SMN2KMT2A
SCHEMBL4874455 0.86 ALDH1A1 (0.76) ALDH1A1LMNAKDM4EKMT2AMEN1
SCHEMBL3840479 0.84 KDM4E (0.56) ALDH1A1KDM4EKMT2AMEN1KDR
Hydrochloric Acid SCHEMBL4873626 0.82 KDM4E (0.55) ALDH1A1KDM4EKMT2AMEN1KDR
SCHEMBL3841498 0.81 KMT2A (0.56) ALDH1A1KDM4EKMT2AMEN1GAA
SCHEMBL4471401 0.80 KDM4E (0.74) ALDH1A1LMNAKDM4EKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1553092-B1 ARALKYL FORMYL-ALKYL PIPERAZINE DERIVATIVES AND THEIR USES AS CEREBRAL NERVE PROTECTIVE AGENT SHANGHAI INST PHARM INDUSTRY (CN) 2009-11-04 EP claimed