SCHEMBL3839017

SCHEMBL3839017

Clc1cccc(OCc2c[nH]cn2)c1Cl.Fc1cccc(OCc2c[nH]cn2)c1F

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MRGPRX4 Q96LA9 2/20 0.39
FFAR1 O14842 1/20 0.38
KDM4E B2RXH2 1/20 0.36
SLC6A2 P23975 3/20 0.36
SLC6A4 P31645 3/20 0.36
SLC6A3 Q01959 3/20 0.36
HTR1A P08908 2/20 0.36
ALDH1A1 P00352 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
HTT P42858 1/20 0.34
TP53 P04637 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
TSHR P16473 1/20 0.33
CYP2C19 P33261 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
RXRA P19793 1/20 0.32
GRIN1 Q05586 1/20 0.32
GRIN2B Q13224 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3834244 0.90 MRGPRX4 (0.35) MRGPRX4FFAR1KDM4ESLC6A2SLC6A4
SCHEMBL222798 0.89 MRGPRX4 (0.46) MRGPRX4KDM4EALDH1A1SMN1; SMN2HTT
SCHEMBL223728 0.89 FFAR1 (0.44) MRGPRX4FFAR1SLC6A2SLC6A4SLC6A3
SCHEMBL3836799 0.82 TP53 (0.40) MRGPRX4FFAR1KDM4EALDH1A1SMN1; SMN2
SCHEMBL3839020 0.81 FFAR1 (0.40) MRGPRX4FFAR1KDM4ESLC6A2SLC6A4
SCHEMBL224611 0.78 TP53 (0.45) FFAR1KDM4EALDH1A1SMN1; SMN2HTT
SCHEMBL224876 0.78 MEN1 (0.44) MRGPRX4FFAR1KDM4EALDH1A1CYP1A2
SCHEMBL6358732 0.73 ALDH1A1 (0.38) HTR1AALDH1A1SMN1; SMN2MAPK14
SCHEMBL2103277 0.70 TAAR1 (0.45) KDM4ESMN1; SMN2HTTCYP1A2CYP3A4
SCHEMBL224383 0.68 HRH3 (0.40) FFAR1SLC6A4HTR1ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2094668-A2 4-IMIDAZOLINES AS TAAR'S LIGANDS F. Hoffmann-Roche AG (CH) 2009-09-02 EP disclosed
WO-2008074679-A2 4-IMIDAZOLINES AS TAAR'S LIGANDS F. HOFFMANN-LA ROCHE AG (CH) 2008-06-26 WO disclosed