SCHEMBL3836799

SCHEMBL3836799

Clc1ccccc1OCc1c[nH]cn1.Fc1ccccc1OCc1c[nH]cn1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 2/20 0.40
HTT P42858 1/20 0.40
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
CYP1A2 P05177 3/20 0.39
CYP2D6 P10635 3/20 0.39
CYP2C19 P33261 3/20 0.39
CYP2C9 P11712 2/20 0.39
RECQL P46063 1/20 0.39
FFAR1 O14842 2/20 0.38
DAO P14920 1/20 0.38
L3MBTL1 Q9Y468 4/20 0.38
TDP1 Q9NUW8 1/20 0.38
NPC1 O15118 3/20 0.37
RAB9A P51151 3/20 0.37
SMN1; SMN2 Q16637 3/20 0.37
HPGD P15428 3/20 0.37
KDM4E B2RXH2 2/20 0.37
MRGPRX4 Q96LA9 1/20 0.37
MAPT P10636 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL224611 0.91 TP53 (0.45) TP53HTTMEN1KMT2ACYP1A2
SCHEMBL224876 0.91 MEN1 (0.44) MEN1KMT2ACYP1A2CYP2D6CYP2C19
SCHEMBL3839017 0.82 MRGPRX4 (0.39) TP53HTTCYP1A2CYP2D6CYP2C19
SCHEMBL6358732 0.80 ALDH1A1 (0.38) MEN1KMT2AL3MBTL1NPC1RAB9A
SCHEMBL222798 0.80 MRGPRX4 (0.46) TP53HTTMEN1KMT2ACYP1A2
SCHEMBL223728 0.80 FFAR1 (0.44) MEN1KMT2ACYP1A2CYP2D6CYP2C19
SCHEMBL3836804 0.80 FFAR1 (0.40) TP53HTTMEN1KMT2AFFAR1
SCHEMBL3834244 0.74 MRGPRX4 (0.35) MEN1KMT2AFFAR1L3MBTL1TDP1
SCHEMBL223566 0.73 ALDH1A1 (0.50) MEN1KMT2ACYP1A2CYP2D6CYP2C19
SCHEMBL224554 0.73 LTA4H (0.50) L3MBTL1TDP1MAPTMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2094668-A2 4-IMIDAZOLINES AS TAAR'S LIGANDS F. Hoffmann-Roche AG (CH) 2009-09-02 EP disclosed
WO-2008074679-A2 4-IMIDAZOLINES AS TAAR'S LIGANDS F. HOFFMANN-LA ROCHE AG (CH) 2008-06-26 WO disclosed