SCHEMBL3839121

SCHEMBL3839121

CC(C)CNCc1cc2c(c(-c3cc4cc(CN5CCCCC5)ccc4[nH]3)c1)C(=O)NC2

nearest known ligand 0.48

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 14/20 0.48
AURKA O14965 6/20 0.46
KDR P35968 6/20 0.46
CDK1 P06493 1/20 0.39
CDK7 P50613 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3887530 0.85 AURKA (0.49) CHEK1AURKAKDR
SCHEMBL3839118 0.84 CHEK1 (0.49) CHEK1AURKAKDRCDK1CDK7
SCHEMBL3837181 0.82 CHEK1 (0.56) CHEK1AURKAKDRCDK1CDK7
Hydrochloric Acid SCHEMBL3874594 0.82 CHEK1 (0.49) CHEK1AURKAKDRCDK1
SCHEMBL3839156 0.81 CHEK1 (0.56) CHEK1AURKAKDRCDK1CDK7
SCHEMBL3839022 0.81 CHEK1 (0.63) CHEK1AURKAKDRCDK1CDK7
Hydrochloric Acid SCHEMBL3841238 0.81 CHEK1 (0.49) CHEK1AURKAKDRCDK1CDK7
Hydrochloric Acid SCHEMBL3837129 0.80 CHEK1 (0.47) CHEK1AURKAKDRCDK1
SCHEMBL3887524 0.79 KDR (0.49) CHEK1AURKAKDR
Hydrochloric Acid SCHEMBL3837133 0.79 CHEK1 (0.47) CHEK1AURKAKDRCDK1CDK7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2108642-A1 JAK INHIBITOR Kyowa Hakko Kirin Co., Ltd. (JP) 2009-10-14 EP disclosed