SCHEMBL3839296

SCHEMBL3839296

CC(C)(C)OC(=O)Nc1cccc(-c2ccc(I)c3c2CNC3=O)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.48
CREBBP Q92793 1/20 0.48
KDR P35968 16/20 0.46
CYP17A1 P05093 1/20 0.44
RIPK3 Q9Y572 2/20 0.42
ROCK2 O75116 3/20 0.41
RET P07949 3/20 0.41
AURKB Q96GD4 3/20 0.41
FLT1 P17948 2/20 0.41
EPHA2 P29317 2/20 0.41
FLT4 P35916 2/20 0.41
FLT3 P36888 2/20 0.41
MAP4K4 O95819 2/20 0.41
LCK P06239 2/20 0.41
PIM1 P11309 2/20 0.41
RPS6KB1 P23443 2/20 0.41
BLK P51451 2/20 0.41
STK3 Q13188 2/20 0.41
ROCK1 Q13464 2/20 0.41
NTRK3 Q16288 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3836940 0.88 KDR (0.60) BRD4CREBBPKDRCYP17A1RIPK3
SCHEMBL3039531 0.72 KDR (0.34) KDRPIM1ROCK1CLK4
SCHEMBL3835838 0.72 TDP2 (0.42) BRD4CREBBPKDRMAP4K4
SCHEMBL3039949 0.71 MAP3K9 (0.50) KDRPIM1ROCK1PRKD3NTRK2
SCHEMBL3840842 0.70 KDR (0.71) KDRROCK2RETAURKBFLT1
SCHEMBL13754832 0.70 CYP17A1 (0.64) BRD4CREBBPCYP17A1
SCHEMBL18170628 0.70 KDR (0.70) KDRROCK2RETAURKBFLT1
SCHEMBL29029431 0.69 HDAC3 (0.56) BRD4CREBBPCYP17A1
SCHEMBL3785736 0.69 BRD4 (0.53) BRD4CREBBPCYP17A1MAP4K4
SCHEMBL5846227 0.69 GPR119 (0.53) BRD4CREBBPCYP17A1NTRK2CLK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2108642-A1 JAK INHIBITOR Kyowa Hakko Kirin Co., Ltd. (JP) 2009-10-14 EP disclosed