SCHEMBL3841864

SCHEMBL3841864

CN(C)Cc1c(Cl)ccc(O)c1Cl

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.48
MAPK1 P28482 2/20 0.48
KDM4E B2RXH2 4/20 0.46
TDP1 Q9NUW8 3/20 0.46
MAPT P10636 2/20 0.46
ALDH1A1 P00352 5/20 0.45
GAA P10253 3/20 0.45
MEN1 O00255 1/20 0.45
POLB P06746 1/20 0.45
THRB P10828 1/20 0.45
G6PD P11413 1/20 0.45
PABPC1 P11940 1/20 0.45
KMT2A Q03164 1/20 0.45
HKDC1 Q2TB90 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
ADRB2 P07550 1/20 0.40
PKM P14618 1/20 0.40
HSD17B10 Q99714 3/20 0.37
TSHR P16473 3/20 0.37
GLA P06280 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8392135 0.86 KDM4E (0.49) CYP3A4MAPK1KDM4ETDP1MAPT
SCHEMBL8388479 0.78 KDM4E (0.49) KDM4ETDP1MAPTALDH1A1GAA
SCHEMBL27695109 0.76 CYP3A4 (0.54) CYP3A4MAPK1TDP1ALDH1A1HSD17B10
SCHEMBL22048288 0.73 SLC6A2 (0.46) CYP3A4MAPTALDH1A1GAAPOLB
SCHEMBL28985928 0.72 CYP3A4 (0.50) CYP3A4MAPK1TDP1ALDH1A1HSD17B10
SCHEMBL9389821 0.71 CYP3A4 (0.54) CYP3A4MAPK1TDP1MAPTALDH1A1
SCHEMBL11653027 0.69 HIF1A (0.63) CYP3A4MAPK1KDM4ETDP1MAPT
SCHEMBL8772350 0.69 CA2 (0.52) CYP3A4KDM4ETDP1MAPTALDH1A1
SCHEMBL7109825 0.69 MAPT (0.57) CYP3A4MAPK1KDM4ETDP1MAPT
SCHEMBL8389821 0.68 ALDH1A1 (0.71) MAPK1KDM4ETDP1MAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2088861-A2 BENZIMIDAZOLE COMPOUNDS Takeda Pharmaceutical Company Limited (JP) 2009-08-19 EP disclosed
WO-2008051533-A2 BENZIMIDAZOLE COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-05-02 WO disclosed