SCHEMBL3844258

SCHEMBL3844258

O=C(O)Cc1cc(Br)c[nH]c1=O

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERCC1 P07992 1/20 0.50
ERCC4 Q92889 1/20 0.50
TSHR P16473 2/20 0.39
ALDH1A1 P00352 2/20 0.39
LMNA P02545 1/20 0.39
GLA P06280 1/20 0.39
CYP2C9 P11712 1/20 0.39
HPGD P15428 1/20 0.39
NFKB1 P19838 1/20 0.39
PMP22 Q01453 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
DAO P14920 1/20 0.37
CREBBP Q92793 1/20 0.37
GRIN2D O15399 1/20 0.37
GRIN3B O60391 1/20 0.37
GRIN1 Q05586 1/20 0.37
GRIN2A Q12879 1/20 0.37
GRIN2B Q13224 1/20 0.37
GRIN2C Q14957 1/20 0.37
GRIN3A Q8TCU5 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13729262 0.80 CREBBP (0.47) ERCC1ERCC4CYP2C9CREBBPGRIN2D
SCHEMBL15228262 0.80 ERCC1 (0.44) ERCC1ERCC4TSHRALDH1A1GLA
SCHEMBL1921613 0.77 KMT2A (0.54) ERCC1ERCC4ALDH1A1LMNAHPGD
SCHEMBL17546137 0.76 ERCC1 (0.52) ERCC1ERCC4TSHRALDH1A1LMNA
SCHEMBL3843553 0.75 ERCC1 (0.43) ERCC1ERCC4TSHRALDH1A1HPGD
SCHEMBL10816643 0.75 ALDH1A1 (0.42) ERCC1ERCC4TSHRALDH1A1LMNA
SCHEMBL25420774 0.72 EPHX2 (0.51) ERCC1ERCC4TSHRALDH1A1GLA
SCHEMBL4725368 0.71 DYRK1A (0.60) ERCC1ERCC4ALDH1A1GLAHPGD
SCHEMBL3637120 0.70 CSNK2A1 (0.46) ERCC1ERCC4ALDH1A1GLAHPGD
SCHEMBL2351513 0.68 AURKA (0.45) TSHRLMNAHPGDMAPTAKR1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018193387-A1 HETEROCYCLIC COMPOUNDS WITH MICROBIOCIDAL PROPERTIES PI INDUSTRIES LTD. (IN) 2018-10-25 WO disclosed
EP-2114898-A2 NITROGEN-CONTAINING HETEROCYCLYL KETONES AND THEIR USE AS C-MET INHIBITORS Amgen Inc. (US) 2009-11-11 EP disclosed
WO-2008103277-A2 NITROGEN-CONTAINING HETEROCYCLYL KETONES AND THEIR USE AS C-MET INHIBITORS AMGEN INC. (US) 2008-08-28 WO disclosed