SCHEMBL3845874

SCHEMBL3845874

Fc1ccc(-c2nn(C(c3ccccc3)(c3ccccc3)c3ccccc3)cc2-c2ccc3ncn(-c4ccc(Cl)cn4)c3c2)c(F)c1

nearest known ligand 0.35

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CDK9 P50750 15/20 0.34
ATM Q13315 1/20 0.32
ALDH1A1 P00352 1/20 0.31
MAPT P10636 1/20 0.31
GRM2 Q14416 1/20 0.31
FGFR1 P11362 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3850334 0.92 ALDH1A1 (0.38) CDK9ATMALDH1A1MAPTFGFR1
SCHEMBL3853393 0.89 MAPK14 (0.32) CDK9ALDH1A1MAPT
SCHEMBL3845877 0.85
SCHEMBL3854592 0.82 FGFR1 (0.35) ALDH1A1MAPTFGFR1
SCHEMBL3849277 0.80 JAK2 (0.35) CDK9FGFR1
SCHEMBL3847147 0.80 FGFR1 (0.39) ALDH1A1MAPTFGFR1
SCHEMBL3846713 0.80 POLB (0.41) CDK9
SCHEMBL5852255 0.78 SRC (0.38) ATMALDH1A1MAPTFGFR1
Hydrochloric Acid SCHEMBL3847696 0.77 ATM (0.34) CDK9ATMGRM2
SCHEMBL3850336 0.77 ALDH1A1 (0.34) ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2048142-A2 Nitrogen-containing condensed cyclic compound having a pyrazolyl group as a substituent group and pharmaceutical composition thereof Eisai R&D Management Co., Ltd. (JP) 2009-04-15 EP disclosed
EP-1382603-B1 NITROGENOUS FUSED-RING COMPOUND HAVING PYRAZOLYL GROUP AS SUBSTITUENT AND MEDICINAL COMPOSITION THEREOF EISAI R&D MAN CO LTD (JP) 2008-07-23 EP disclosed
US-7074801-B1 Nitrogen-containing condensed cyclic compound having a pyrazolyl group as a substituent group and pharmaceutical composition thereof EISAI CO., LTD. (JP) 2006-07-11 US disclosed
EP-1382603-A1 NITROGENOUS FUSED−RING COMPOUND HAVING PYRAZOLYL GROUP AS SUBSTITUENT AND MEDICINAL COMPOSITION THEREOF Eisai Co., Ltd. (JP) 2004-01-21 EP disclosed