SCHEMBL3846110

SCHEMBL3846110

O=C(Nc1cccc(F)c1F)c1ccc(-c2cnc3ccc(-c4cn[nH]c4)cn23)cc1F

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
FLT3 P36888 2/20 0.44
NRAS P01111 1/20 0.44
ROCK2 O75116 5/20 0.42
ROCK1 Q13464 4/20 0.42
CHEK1 O14757 9/20 0.41
CHEK2 O96017 3/20 0.41
ABL1 P00519 1/20 0.40
KIT P10721 1/20 0.40
PTK6 Q13882 1/20 0.39
AURKB Q96GD4 1/20 0.39
MAPK1 P28482 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5854241 0.99 FLT3 (0.43) FLT3NRASROCK2ROCK1CHEK1
SCHEMBL3854844 0.87 FLT3 (0.42) FLT3NRASROCK2ROCK1CHEK1
SCHEMBL4712318 0.87 KDM4E (0.41) FLT3NRASROCK2ROCK1CHEK1
Hydrochloric Acid SCHEMBL5853292 0.86 FLT3 (0.42) FLT3NRASROCK2ROCK1CHEK1
Hydrochloric Acid SCHEMBL3849122 0.86 KDM4E (0.40) FLT3NRASROCK2ROCK1CHEK1
Hydrochloric Acid SCHEMBL3847703 0.85 ROCK2 (0.44) FLT3NRASROCK2ROCK1CHEK1
Hydrochloric Acid SCHEMBL3846279 0.85 MET (0.42) FLT3NRASROCK2ROCK1CHEK1
Hydrochloric Acid SCHEMBL3846953 0.84 KIT (0.39) FLT3NRASROCK2ROCK1CHEK1
Hydrochloric Acid SCHEMBL3845647 0.84 LRRK2 (0.45) FLT3NRASROCK2ROCK1PTK6
Hydrochloric Acid SCHEMBL3849166 0.82 FLT3 (0.42) FLT3NRASROCK2ROCK1CHEK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2048142-A2 Nitrogen-containing condensed cyclic compound having a pyrazolyl group as a substituent group and pharmaceutical composition thereof Eisai R&D Management Co., Ltd. (JP) 2009-04-15 EP disclosed
EP-1382603-B1 NITROGENOUS FUSED-RING COMPOUND HAVING PYRAZOLYL GROUP AS SUBSTITUENT AND MEDICINAL COMPOSITION THEREOF EISAI R&D MAN CO LTD (JP) 2008-07-23 EP disclosed