SCHEMBL3846632

SCHEMBL3846632

CC(C)(C)OC(=O)N1CCN(c2ccc3c(c2)OCO3)CC1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCD5 Q86SK9 1/20 0.58
MAPT P10636 5/20 0.55
ALDH1A1 P00352 3/20 0.55
LMNA P02545 2/20 0.55
KMT2A Q03164 3/20 0.53
PDK2 Q15119 1/20 0.51
TSHR P16473 2/20 0.50
GPR183 P32249 1/20 0.50
GPR119 Q8TDV5 4/20 0.49
GFER P55789 1/20 0.49
HSD17B10 Q99714 1/20 0.49
HTT P42858 1/20 0.48
NAMPT P43490 1/20 0.48
POLB P06746 1/20 0.48
KDM4E B2RXH2 1/20 0.47
MEN1 O00255 1/20 0.47
GAA P10253 1/20 0.47
THRB P10828 1/20 0.47
ALOX15 P16050 1/20 0.47
ALOX12 P18054 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5231045 0.88 MAPT (0.51) SCD5MAPTALDH1A1LMNAKMT2A
SCHEMBL8288524 0.82 ALDH1A1 (0.67) SCD5ALDH1A1LMNAKMT2ATSHR
SCHEMBL5573222 0.82 MAPT (0.76) MAPTALDH1A1LMNAKMT2APDK2
SCHEMBL15979567 0.81 MAPT (0.67) MAPTALDH1A1LMNAKMT2ATSHR
SCHEMBL12208580 0.80 MAPT (0.50) MAPTALDH1A1LMNAKMT2APDK2
SCHEMBL15266373 0.79 SCD5 (0.55) SCD5MAPTALDH1A1GPR183HTT
SCHEMBL3595243 0.79 ALDH1A1 (0.63) MAPTALDH1A1LMNAKMT2AHTT
SCHEMBL5727630 0.79 MAPT (0.49) MAPTALDH1A1LMNAKMT2APDK2
SCHEMBL25447362 0.79 MAPT (0.60) MAPTALDH1A1LMNAKMT2APDK2
SCHEMBL12478533 0.79 DRD2 (0.50) SCD5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250214977-A1 STAT6 INHIBITORS AND USES THEREOF KYMERA THERAPEUTICS, INC. 2025-07-03 US disclosed
CN-116640122-A IKZF 2 Degradation agent, pharmaceutical composition containing degradation agent and application of degradation agent 苏州国匡医药科技有限公司 2023-08-25 CN disclosed
WO-2023155710-A1 IKZF2 DEGRADATION AGENT, PHARMACEUTICAL COMPOSITION COMPRISING SAME AND USE THEREOF 苏州国匡医药科技有限公司 2023-08-24 WO disclosed
EP-2733144-B1 NOVEL COMPOUND HAVING PARP INHIBITORY ACTIVITY SANTEN PHARMACEUTICAL CO LTD (JP) 2016-01-06 EP disclosed
US-9062061-B2 Compound having PARP inhibitory activity SANTEN PHARMACEUTICAL CO., LTD. (JP) 2015-06-23 US disclosed
US-20140243320-A1 NOVEL COMPOUND HAVING PARP INHIBITORY ACTIVITY SANTEN PHARMACEUTICAL CO., LTD. (JP) 2014-08-28 US disclosed
EP-2733144-A1 NOVEL COMPOUND HAVING PARP INHIBITORY ACTIVITY Santen Pharmaceutical Co., Ltd (JP) 2014-05-21 EP disclosed
EP-2048142-A2 Nitrogen-containing condensed cyclic compound having a pyrazolyl group as a substituent group and pharmaceutical composition thereof Eisai R&D Management Co., Ltd. (JP) 2009-04-15 EP disclosed
EP-1382603-B1 NITROGENOUS FUSED-RING COMPOUND HAVING PYRAZOLYL GROUP AS SUBSTITUENT AND MEDICINAL COMPOSITION THEREOF EISAI R&D MAN CO LTD (JP) 2008-07-23 EP disclosed
US-7074801-B1 Nitrogen-containing condensed cyclic compound having a pyrazolyl group as a substituent group and pharmaceutical composition thereof EISAI CO., LTD. (JP) 2006-07-11 US disclosed
EP-1382603-A1 NITROGENOUS FUSED−RING COMPOUND HAVING PYRAZOLYL GROUP AS SUBSTITUENT AND MEDICINAL COMPOSITION THEREOF Eisai Co., Ltd. (JP) 2004-01-21 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140243320-A1 NOVEL COMPOUND HAVING PARP INHIBITORY ACTIVITY PARP1, PARP11, PARP2 SCD5 4152/4885MAPT 3412/4885ALDH1A1 532/4885
US-20250214977-A1 STAT6 INHIBITORS AND USES THEREOF STAT6, STAT5B, STAT5A SCD5 1513/4885MAPT 3335/4885ALDH1A1 3523/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.