SCHEMBL3846763

SCHEMBL3846763

CCSc1nc2ccc(-c3cn(C(c4ccccc4)(c4ccccc4)C4C=CC=CC4)nc3-c3ccc(F)cc3)cc2n1-c1ccc(F)cc1

nearest known ligand 0.32

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.32
PDE7A Q13946 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3848529 0.87 PTGS2 (0.30)
SCHEMBL3855066 0.87 ALDH1A1 (0.32) ALDH1A1
SCHEMBL3852642 0.86 NPSR1 (0.32) ALDH1A1
SCHEMBL3846760 0.84 PDE7A (0.36) ALDH1A1PDE7A
SCHEMBL3850581 0.83 AKT1 (0.33) ALDH1A1
SCHEMBL3847469 0.81
SCHEMBL5852256 0.81 ATM (0.32) ALDH1A1
SCHEMBL3847835 0.76 ALOX5AP (0.37) ALDH1A1
SCHEMBL3846716 0.76 POLB (0.33)
SCHEMBL3846131 0.76 MEN1 (0.38) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2048142-A2 Nitrogen-containing condensed cyclic compound having a pyrazolyl group as a substituent group and pharmaceutical composition thereof Eisai R&D Management Co., Ltd. (JP) 2009-04-15 EP disclosed
EP-1382603-B1 NITROGENOUS FUSED-RING COMPOUND HAVING PYRAZOLYL GROUP AS SUBSTITUENT AND MEDICINAL COMPOSITION THEREOF EISAI R&D MAN CO LTD (JP) 2008-07-23 EP disclosed
US-7074801-B1 Nitrogen-containing condensed cyclic compound having a pyrazolyl group as a substituent group and pharmaceutical composition thereof EISAI CO., LTD. (JP) 2006-07-11 US disclosed
EP-1382603-A1 NITROGENOUS FUSED−RING COMPOUND HAVING PYRAZOLYL GROUP AS SUBSTITUENT AND MEDICINAL COMPOSITION THEREOF Eisai Co., Ltd. (JP) 2004-01-21 EP disclosed