SCHEMBL3847537

SCHEMBL3847537

COc1ccc(CCN2CCC(CCNc3ccc(-c4ccccc4)cc3)CC2)cc1OC.COc1ccc(CCN2CCC(CCNc3ccc4c(c3)OCO4)CC2)cc1OC.COc1ccc(NCCC2CCN(CCc3ccc(OC)c(OC)c3)CC2)cc1

nearest known ligand 0.53

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 2/20 0.47
SLC6A4 P31645 2/20 0.47
ADRA1D P25100 1/20 0.46
ADRA1A P35348 1/20 0.46
ADRA1B P35368 1/20 0.46
ABCB1 P08183 1/20 0.45
LMNA P02545 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
KCNH2 Q12809 1/20 0.44
HTR2A P28223 1/20 0.43
HTR2C P28335 1/20 0.43
HTR2B P41595 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1333195 0.90 ADRA1D (0.50) HTR1ASLC6A4ADRA1DADRA1AADRA1B
SCHEMBL1333252 0.88 ABCB1 (0.56) HTR1ASLC6A4ABCB1
SCHEMBL1333914 0.85 HTR1A (0.59) HTR1ASLC6A4ABCB1KCNH2
SCHEMBL1334517 0.82 ABCB1 (0.60) HTR1ASLC6A4ABCB1
SCHEMBL2567216 0.78 HTR1A (0.53) HTR1ASLC6A4ABCB1
SCHEMBL1332009 0.78 HTR1A (0.52) HTR1ASLC6A4ABCB1
SCHEMBL2574419 0.78 HTR1A (0.52) HTR1ASLC6A4ABCB1
SCHEMBL5276521 0.78 ACHE (0.61) HTR1ASLC6A4
SCHEMBL1334361 0.77 HTR1A (0.55) HTR1ASLC6A4ADRA1DADRA1AADRA1B
SCHEMBL1332119 0.77 HTR1A (0.51) HTR1ASLC6A4ABCB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1978959-A4 PIPERIDINE AND PIPERAZINE DERIVATIVES MS SCIENCE CORP (JP) 2009-09-02 EP disclosed
EP-1978959-A2 PIPERIDINE AND PIPERAZINE DERIVATIVES M's Science Corporation (JP) 2008-10-15 EP disclosed
WO-2008096189-A2 PIPERIDINE AND PIPERAZINE DERIVATIVES M'S SCIENCE CORPORATION (JP) 2008-08-14 WO disclosed