SCHEMBL3847872

SCHEMBL3847872

Cc1csc(NC(=O)c2ccc(-c3cnc4ccc(Br)cn34)cc2)n1

nearest known ligand 0.57

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.57
RAB9A P51151 7/20 0.51
NPC1 O15118 7/20 0.51
KDM4E B2RXH2 2/20 0.51
SMN1; SMN2 Q16637 2/20 0.51
HTT P42858 1/20 0.51
ALDH1A1 P00352 3/20 0.49
HPGD P15428 1/20 0.49
KMT2A Q03164 4/20 0.49
MEN1 O00255 3/20 0.49
GAA P10253 1/20 0.49
SORT1 Q99523 1/20 0.47
TDP1 Q9NUW8 1/20 0.46
PKM P14618 1/20 0.45
CASP3 P42574 1/20 0.45
SENP8 Q96LD8 1/20 0.45
SENP7 Q9BQF6 1/20 0.45
SENP6 Q9GZR1 1/20 0.45
SCD O00767 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL3849378 0.84 MAPT (0.50) MAPTRAB9ANPC1KDM4ESMN1; SMN2
Hydrochloric Acid SCHEMBL3847648 0.82 MAPT (0.48) MAPTRAB9ANPC1KDM4ESMN1; SMN2
SCHEMBL3848191 0.80 NPC1 (0.48) MAPTRAB9ANPC1HTTALDH1A1
SCHEMBL14145116 0.79 ATM (0.63)
SCHEMBL3847053 0.79 NPC1 (0.46) MAPTRAB9ANPC1HTTALDH1A1
SCHEMBL3846567 0.78 NPC1 (0.48) MAPTRAB9ANPC1KDM4ESMN1; SMN2
SCHEMBL3850904 0.77 MAPT (0.49) MAPTRAB9ANPC1SMN1; SMN2KMT2A
SCHEMBL3850100 0.75 PIK3CA (0.53) KDM4EALDH1A1
SCHEMBL3847512 0.73 MKNK1 (0.51) ALDH1A1HPGD
SCHEMBL3846712 0.72 MKNK1 (0.61)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2048142-A2 Nitrogen-containing condensed cyclic compound having a pyrazolyl group as a substituent group and pharmaceutical composition thereof Eisai R&D Management Co., Ltd. (JP) 2009-04-15 EP disclosed
EP-1382603-B1 NITROGENOUS FUSED-RING COMPOUND HAVING PYRAZOLYL GROUP AS SUBSTITUENT AND MEDICINAL COMPOSITION THEREOF EISAI R&D MAN CO LTD (JP) 2008-07-23 EP disclosed
US-7074801-B1 Nitrogen-containing condensed cyclic compound having a pyrazolyl group as a substituent group and pharmaceutical composition thereof EISAI CO., LTD. (JP) 2006-07-11 US disclosed
EP-1382603-A1 NITROGENOUS FUSED−RING COMPOUND HAVING PYRAZOLYL GROUP AS SUBSTITUENT AND MEDICINAL COMPOSITION THEREOF Eisai Co., Ltd. (JP) 2004-01-21 EP disclosed