SCHEMBL3853255

SCHEMBL3853255

Cc1c(-c2ccccc2)ccc(S(N)(=O)=O)c1-c1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 5/20 0.44
CA1 P00915 5/20 0.41
CA2 P00918 5/20 0.41
CA12 O43570 4/20 0.41
CA9 Q16790 4/20 0.41
PTGS2 P35354 4/20 0.39
CA4 P22748 3/20 0.39
CA6 P23280 3/20 0.39
CA5A P35218 2/20 0.39
CA7 P43166 2/20 0.39
CA14 Q9ULX7 2/20 0.39
CA5B Q9Y2D0 2/20 0.39
PTGS1 P23219 2/20 0.39
MT-CO2 P00403 1/20 0.39
LMNA P02545 1/20 0.39
CA3 P07451 1/20 0.39
ADRB2 P07550 1/20 0.39
ADRB1 P08588 1/20 0.39
CYP3A4 P08684 1/20 0.39
ADORA3 P0DMS8 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4073856 0.86 LRRK2 (0.51) LRRK2CA1CA2CA12CA9
SCHEMBL8976123 0.81 CA2 (0.52) CA1CA2CA12CA9PTGS2
SCHEMBL27181150 0.81 CA2 (0.41) CA1CA2CA12CA9PTGS2
SCHEMBL28134095 0.80 MAOB (0.49) CA1CA2CA12CA9PTGS2
SCHEMBL31457100 0.80 CA1 (0.39) LRRK2CA1CA2CA12CA9
SCHEMBL3823919 0.79 CA1 (0.40) LRRK2CA1CA2CA12CA9
SCHEMBL2896796 0.79 LRRK2 (0.51) LRRK2CA1CA2CA12CA9
Hydrochloric Acid SCHEMBL5808148 0.77 MAOB (0.47) LRRK2CA1CA2CA12CA9
SCHEMBL4759798 0.77 CASP1 (0.48) CA1CA2CA12CA9PTGS2
SCHEMBL27895889 0.75 CA2 (0.52) CA1CA2CA12CA9PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2104677-A1 SPIROPIPERIDINE GLYCINAMIDE DERIVATIVES F. Hoffmann-Roche AG (CH) 2009-09-30 EP disclosed
WO-2008084005-A1 SPIROPIPERIDINE GLYCINAMIDE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2008-07-17 WO disclosed