SCHEMBL3854464

SCHEMBL3854464

Cc1cc(NC(=O)c2ccc3c(c2)CCN(C(=O)O)C3C(C)(C)C)nn1Cc1ccccc1-c1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PTGER1 P34995 15/20 0.42
KMT2A Q03164 1/20 0.36
KCNA5 P22460 1/20 0.35
KCNH2 Q12809 1/20 0.35
TP53 P04637 1/20 0.35
LMNA P02545 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
TSHR P16473 1/20 0.35
CYP2C19 P33261 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
HSD17B10 Q99714 1/20 0.35
NPC1 O15118 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3847522 0.89 PTGER1 (0.45) PTGER1KMT2ALMNACYP1A2CYP3A4
SCHEMBL3854465 0.86 PTGER1 (0.46) PTGER1
SCHEMBL3856743 0.84 PTGER1 (0.46) PTGER1KMT2ATP53LMNATSHR
SCHEMBL4795243 0.79 PTGER1 (0.70) PTGER1
SCHEMBL3186192 0.79 PTGER1 (0.48) PTGER1
SCHEMBL3180838 0.77 PTGER1 (0.61) PTGER1KMT2ACYP3A4
Hydrochloric Acid SCHEMBL3187915 0.76 PTGER1 (0.61) PTGER1CYP3A4
SCHEMBL3847525 0.75 PTGER1 (0.48) PTGER1
SCHEMBL3176032 0.71 PTGER1 (0.67) PTGER1LMNACYP1A2CYP3A4CYP2D6
SCHEMBL3179276 0.71 PTGER1 (0.65) PTGER1TP53LMNACYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2106398-A2 ISOQUINOLINECARBOXAMIDES AS INHIBITORS OF STEAROYL-COA DESATURASE (SCD) SmithKline Beecham Corporation (US) 2009-10-07 EP disclosed
WO-2008074832-A2 ISOQUINOLINECARBOXAMIDES AS INHIBITORS OF STEAROYL-COA DESATURASE ( SCD) SMITHKLINE BEECHAM CORPORATION (US) 2008-06-26 WO disclosed