SCHEMBL3847522

SCHEMBL3847522

COc1ccccc1Cn1nc(NC(=O)c2ccc3c(c2)CCN(C(=O)O)C3C(C)(C)C)cc1C

nearest known ligand 0.45

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PTGER1 P34995 13/20 0.45
LMNA P02545 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
TSHR P16473 1/20 0.40
CYP2C19 P33261 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
HSD17B10 Q99714 1/20 0.40
MAPT P10636 1/20 0.39
KMT2A Q03164 2/20 0.38
NPC1 O15118 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3854464 0.89 PTGER1 (0.42) PTGER1LMNACYP1A2CYP3A4CYP2D6
SCHEMBL3847525 0.87 PTGER1 (0.48) PTGER1
SCHEMBL3856743 0.83 PTGER1 (0.46) PTGER1LMNATSHRSMN1; SMN2HSD17B10
SCHEMBL4795243 0.82 PTGER1 (0.70) PTGER1
SCHEMBL3587201 0.79 PTGER1 (0.50) PTGER1LMNACYP1A2CYP3A4CYP2D6
SCHEMBL3578786 0.76 PTGER1 (0.65) PTGER1LMNACYP1A2CYP3A4CYP2D6
Hydrochloric Acid SCHEMBL3583491 0.75 PTGER1 (0.66) PTGER1LMNACYP1A2CYP3A4CYP2D6
SCHEMBL3854465 0.75 PTGER1 (0.46) PTGER1
SCHEMBL3581181 0.71 PTGER1 (0.48) PTGER1
SCHEMBL3666730 0.70 KDM1A (0.43) NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2102188-A2 COMPOUNDS SmithKline Beecham Corporation (US) 2009-09-23 EP disclosed
WO-2008074833-A2 COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2008-06-26 WO disclosed