SCHEMBL3856743

SCHEMBL3856743

Cc1cc(NC(=O)c2ccc3c(c2)CCN(C(=O)O)C3C(C)(C)C)nn1Cc1cccc(Cl)c1

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PTGER1 P34995 13/20 0.46
TP53 P04637 1/20 0.44
P2RY14 Q15391 1/20 0.44
LMNA P02545 2/20 0.41
KMT2A Q03164 1/20 0.41
SMN1; SMN2 Q16637 3/20 0.41
TSHR P16473 2/20 0.41
NPSR1 Q6W5P4 2/20 0.41
ALDH1A1 P00352 1/20 0.41
HSD17B10 Q99714 1/20 0.40
MAPT P10636 1/20 0.40
HTT P42858 1/20 0.40
THRB P10828 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3856745 0.86 PTGER1 (0.49) PTGER1TP53P2RY14SMN1; SMN2NPSR1
SCHEMBL3854464 0.84 PTGER1 (0.42) PTGER1TP53LMNAKMT2ASMN1; SMN2
SCHEMBL3847522 0.83 PTGER1 (0.45) PTGER1LMNAKMT2ASMN1; SMN2TSHR
SCHEMBL4795243 0.83 PTGER1 (0.70) PTGER1
SCHEMBL3186899 0.78 PTGER1 (0.52) PTGER1TP53P2RY14LMNAKMT2A
SCHEMBL3177484 0.76 PTGER1 (0.66) PTGER1TP53P2RY14LMNAKMT2A
SCHEMBL4022471 0.76 PTGDR2 (0.39) TP53LMNAKMT2ASMN1; SMN2TSHR
SCHEMBL3844835 0.75 PTGER1 (0.61) PTGER1
SCHEMBL4433371 0.73 PPARA (0.37) LMNASMN1; SMN2ALDH1A1MAPTHTT
SCHEMBL4422304 0.72 GAA (0.54) TP53LMNAKMT2ASMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2106398-A2 ISOQUINOLINECARBOXAMIDES AS INHIBITORS OF STEAROYL-COA DESATURASE (SCD) SmithKline Beecham Corporation (US) 2009-10-07 EP disclosed
WO-2008074832-A2 ISOQUINOLINECARBOXAMIDES AS INHIBITORS OF STEAROYL-COA DESATURASE ( SCD) SMITHKLINE BEECHAM CORPORATION (US) 2008-06-26 WO disclosed