SCHEMBL3860080

SCHEMBL3860080

CC(C)(C)OC(=O)NCCOc1cccc(CC#CCc2ccccc2)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.51
PDK2 Q15119 1/20 0.51
CA12 O43570 3/20 0.49
CA1 P00915 3/20 0.49
CA2 P00918 3/20 0.49
CA9 Q16790 3/20 0.49
MTNR1A P48039 2/20 0.45
MTNR1B P49286 2/20 0.45
BCHE P06276 2/20 0.45
CNR2 P34972 2/20 0.45
L3MBTL1 Q9Y468 2/20 0.44
MAPT P10636 1/20 0.44
NPC1 O15118 1/20 0.44
POLB P06746 1/20 0.44
CASP3 P42574 1/20 0.44
RAB9A P51151 1/20 0.44
SENP7 Q9BQF6 1/20 0.44
MAOB P27338 1/20 0.43
DRD2 P14416 1/20 0.43
DRD4 P21917 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3861248 0.92 CA12 (0.48) IDO1PDK2CA12CA1CA2
SCHEMBL233621 0.90 CA12 (0.49) IDO1PDK2CA12CA1CA2
SCHEMBL31724915 0.85 CA12 (0.52) IDO1PDK2CA12CA1CA2
SCHEMBL28430727 0.85 CA12 (0.52) IDO1PDK2CA12CA1CA2
SCHEMBL17974300 0.84 CA12 (0.54) IDO1PDK2CA12CA1CA2
SCHEMBL3869724 0.84 MTNR1A (0.49) MTNR1AMTNR1BL3MBTL1NPC1POLB
SCHEMBL236856 0.84 CA12 (0.54) IDO1PDK2CA12CA1CA2
SCHEMBL17974302 0.83 CA12 (0.53) IDO1PDK2CA12CA1CA2
SCHEMBL236608 0.83 CA12 (0.47) IDO1PDK2CA12CA1CA2
SCHEMBL23705710 0.83 L3MBTL1 (0.62) IDO1PDK2CA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2076122-A2 ALKYNYL PHENYL DERIVATIVE COMPOUNDS FOR TREATING OPHTHALMIC DISEASES AND DISORDERS Acucela, Inc. (US) 2009-07-08 EP disclosed
WO-2009005794-A2 ALKYNYL PHENYL DERIVATIVE COMPOUNDS FOR TREATING OPHTHALMIC DISEASES AND DISORDERS ACUCELA, INC. (US) 2009-01-08 WO disclosed