Lysine

Lysine

SCHEMBL3868637

NCCCC[C@H](N)C(=O)O.O=C1C=CC(=O)N1

nearest known ligand 0.67

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

PPARDPTGS1PTGS2dacAdacBdacCftsImrcAmrcBmrdA

The experimentally established mechanism targets of Lysine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GSR P00390 1/20 0.67
ARG2 P78540 4/20 0.43
ARG1 P05089 3/20 0.43
ITGB3 P05106 1/20 0.42
ITGA2B P08514 1/20 0.42
RNPEP Q9H4A4 1/20 0.42
POLB P06746 1/20 0.41
KMT2A Q03164 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
CPB2 Q96IY4 2/20 0.40
CPB1 P15086 1/20 0.40
DPP8 Q6V1X1 1/20 0.40
DPP9 Q86TI2 1/20 0.40
DPP7 Q9UHL4 1/20 0.40
THRB P10828 1/20 0.40
AGER Q15109 1/20 0.40
MMP2 P08253 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Lysine SCHEMBL28207112 1.00 GSR (0.67) GSRARG2ARG1ITGB3ITGA2B
Lysine SCHEMBL28860372 0.94 GSR (0.59) GSRARG2ARG1ITGB3ITGA2B
Lysine SCHEMBL28207652 0.87 GSR (0.50) GSRARG2ARG1ITGB3ITGA2B
Lysine SCHEMBL28980840 0.84 GSR (0.74) GSRARG2ARG1RNPEPPOLB
Lysine SCHEMBL28980842 0.84 GSR (0.74) GSRARG2ARG1RNPEPPOLB
Lysine SCHEMBL29075874 0.84 GSR (0.95) GSRARG2ARG1RNPEPCPB2
Norleucine SCHEMBL27512040 0.83 SLC1A2 (0.49) GSRDPP7AGER
Lysine SCHEMBL28214073 0.82 GSR (0.91) GSRARG2ARG1RNPEPPOLB
Lysine SCHEMBL3029499 0.82 GSR (0.91) GSRARG2ARG1RNPEPCPB2
Lysine SCHEMBL1000151 0.82 GSR (1.00) GSRARG2ARG1RNPEPKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 24 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12029733-B2 Treatment of sepsis and related inflammatory conditions by local neuromodulation of the autonomic nervous system Tulavi Therapeutics, Inc. (US) 2024-07-09 US disclosed
US-11446359-B2 Systems and methods for cardiac plexus neuromodulation Tulavi Therapeutics, Inc. (US) 2022-09-20 US disclosed
US-11154547-B2 Treatment of sepsis and related inflammatory conditions by local neuromodulation of the autonomic nervous system Tulavi Therapeutics, Inc. (US) 2021-10-26 US disclosed
US-20210205501-A1 SYSTEMS AND METHODS FOR GEL-BASED NEUROMODULATION Tulavi Therapeutics, Inc. 2021-07-08 US disclosed
CN-109675020-B Oral GLP-1 polypeptide nano preparation and preparation method and application thereof 浙江大学 2021-05-04 CN disclosed
EP-3764990-A1 SYSTEMS AND METHODS FOR GEL-BASED NEUROMODULATION Tulavi Therapeutics, Inc. (US) 2021-01-20 EP disclosed
CN-112118828-A Systems and methods for gel-based neuromodulation 图拉维治疗股份有限公司 2020-12-22 CN disclosed
US-20200085809-A1 TREATMENT OF SEPSIS AND RELATED INFLAMMATORY CONDITIONS BY LOCAL NEUROMODULATION OF THE AUTONOMIC NERVOUS SYSTEM Tulavi Therapeutics, Inc. 2020-03-19 US disclosed
WO-2019178564-A1 SYSTEMS AND METHODS FOR GEL-BASED NEUROMODULATION Tulavi Therapeutics, Inc. (US) 2019-09-19 WO disclosed
CN-110035754-A Pass through the local nerve adjustment for the treatment of septicemia and the related inflammatory patient's condition of autonomic nerves system 图拉维治疗股份有限公司 2019-07-19 CN disclosed
EP-3288626-A1 SYSTEMS AND MEHTODS FOR SYMPATHETIC CARDIOPULMONARY NEUROMODULATION Reflex Medical Inc. (US) 2018-03-07 EP disclosed
WO-2018005848-A1 TREATMENT OF SEPSIS AND RELATED INFLAMMATORY CONDITIONS BY LOCAL NEUROMODULATION OF THE AUTONOMIC NERVOUS SYSTEM BRIGHT, CORINNE (US) 2018-01-04 WO disclosed
US-9855317-B2 Systems and methods for sympathetic cardiopulmonary neuromodulation Reflex Medical, Inc. (US) 2018-01-02 US disclosed
US-20160317621-A1 SYSTEMS AND METHODS FOR SYMPATHETIC CARDIOPULMONARY NEUROMODULATION Tulavi Therapeutics, Inc. 2016-11-03 US disclosed
WO-2016176333-A1 SYSTEMS AND MEHTODS FOR SYMPATHETIC CARDIOPULMONARY NEUROMODULATION Reflex Medical, Inc. (US) 2016-11-03 WO disclosed
US-7595198-B2 Photocleavable isotope-coded affinity tags AMBERGEN, INC. (US) 2009-09-29 US disclosed
US-20080032417-A1 Photocleavable isotope-coded affinity tags AMBERGEN, INC 2008-02-07 US disclosed
US-7145019-B2 Photocleavable isotope-coded affinity tags AMBERGEN, INC. (US) 2006-12-05 US disclosed
WO-2005037210-A2 PHOTOCLEAVABLE ISOTOPE-CODED AFFINITY TAGS AMBERGEN, INC. (US) 2005-04-28 WO disclosed
US-20050085630-A1 Photocleavable isotope-coded affinity tags AMBERGEN INC. 2005-04-21 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050085630-A1 Photocleavable isotope-coded affinity tags PTMS, DNPEP, ACP1 GSR 3944/4885ARG2 4651/4885ARG1 4623/4885
US-20080032417-A1 Photocleavable isotope-coded affinity tags PTMS, DNPEP, ACP1 GSR 3944/4885ARG2 4651/4885ARG1 4623/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.