SCHEMBL3870053

SCHEMBL3870053

O=C1NCC(Cc2ccccc2)N1C1CCN(Cc2ccccc2)CC1

nearest known ligand 0.55

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
OPRL1 P41146 4/20 0.55
CCR3 P51677 1/20 0.52
DRD2 P14416 7/20 0.50
DRD4 P21917 7/20 0.50
DRD3 P35462 7/20 0.50
OPRM1 P35372 3/20 0.50
OPRK1 P41145 2/20 0.50
CHRM3 P20309 4/20 0.48
CHRM2 P08172 3/20 0.48
ALDH1A1 P00352 1/20 0.47
ACHE P22303 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Lithium Ion SCHEMBL3864715 0.96 OPRL1 (0.52) OPRL1CCR3DRD2DRD4DRD3
SCHEMBL3703348 0.83 OPRL1 (0.56) OPRL1DRD2DRD4DRD3OPRM1
SCHEMBL3861071 0.82 GBA1 (0.49)
SCHEMBL3063295 0.78 CHRM3 (0.59) OPRL1DRD2DRD4DRD3OPRM1
SCHEMBL11217794 0.76 OPRL1 (0.57) OPRL1DRD2DRD4DRD3OPRM1
SCHEMBL13986107 0.74 EHMT2 (0.46)
SCHEMBL12614026 0.73 HTR3A (0.41) DRD3OPRM1CHRM2
SCHEMBL3073412 0.71 OPRL1 (0.60) OPRL1CCR3DRD2DRD4DRD3
SCHEMBL31437068 0.71 CHRM3 (0.61) OPRL1DRD2DRD4DRD3OPRM1
SCHEMBL3248256 0.71 CHRM3 (0.54) OPRL1CCR3DRD2DRD4DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1856100-A4 CGRP RECEPTOR ANTAGONISTS MERCK & CO INC (US) 2009-04-15 EP disclosed
EP-1856100-A2 CGRP RECEPTOR ANTAGONISTS Merck & Co., Inc. (US) 2007-11-21 EP disclosed
WO-2006078554-A2 CGRP RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 2006-07-27 WO disclosed