SCHEMBL3876573

SCHEMBL3876573

CCOC(=O)c1cc(CC#N)cnc1N1CCNCC1

nearest known ligand 0.53

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.53
NMT2 O60551 2/20 0.46
NMT1 P30419 2/20 0.46
OPRK1 P41145 6/20 0.45
L3MBTL1 Q9Y468 3/20 0.44
DYRK1A Q13627 1/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
KDM4E B2RXH2 3/20 0.40
LMNA P02545 2/20 0.40
HPGD P15428 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
TP53 P04637 1/20 0.40
HTT P42858 1/20 0.40
ADORA3 P0DMS8 1/20 0.40
PAK1 Q13153 1/20 0.40
MAPT P10636 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3926411 0.81 OPRK1 (0.56) ALDH1A1OPRK1DYRK1AMEN1KMT2A
SCHEMBL21171822 0.78 OPRK1 (0.57) OPRK1MEN1KMT2AKDM4E
SCHEMBL29501650 0.77 KDM4E (0.49) ALDH1A1NMT1L3MBTL1KMT2AKDM4E
SCHEMBL25255731 0.77 KDM4E (0.49) ALDH1A1NMT1L3MBTL1KMT2AKDM4E
SCHEMBL14598715 0.76 ALDH1A1 (0.69) ALDH1A1L3MBTL1MEN1KMT2AKDM4E
SCHEMBL907923 0.74 P2RY12 (0.49) ALDH1A1
SCHEMBL3874439 0.73 ALDH1A1 (0.76) ALDH1A1L3MBTL1MEN1KMT2AKDM4E
SCHEMBL30999840 0.73 ALDH1A1 (0.76) ALDH1A1L3MBTL1MEN1KMT2AKDM4E
SCHEMBL2454645 0.73 OPRK1 (0.57) ALDH1A1OPRK1KMT2ALMNAADORA3
SCHEMBL10516498 0.73 ALDH1A1 (0.51) ALDH1A1NMT2NMT1L3MBTL1DYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2041115-A1 NEW PYRIDINE ANALOGUES AstraZeneca AB (SE) 2009-04-01 EP disclosed
WO-2008004942-A1 NEW PYRIDINE ANALOGUES ASTRAZENECA AB (SE) 2008-01-10 WO disclosed