SCHEMBL3877266

SCHEMBL3877266

CC#CCn1c(=O)n(C)c2ccnc(N3CCN(C(=O)OC(C)(C)C)CC3)c21

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ACHE P22303 2/20 0.40
GPR119 Q8TDV5 5/20 0.40
GRIA1 P42261 1/20 0.39
KIT P10721 2/20 0.38
AOC3 Q16853 1/20 0.38
RET P07949 1/20 0.38
POLB P06746 1/20 0.37
DDB1 Q16531 1/20 0.37
CRBN Q96SW2 1/20 0.37
CKS1B P61024 1/20 0.37
SKP1 P63208 1/20 0.37
SKP2 Q13309 1/20 0.37
DPP4 P27487 1/20 0.37
MMP1 P03956 1/20 0.37
MMP13 P45452 1/20 0.37
ADAM17 P78536 1/20 0.37
PDE10A Q9Y233 1/20 0.37
DTYMK P23919 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13876175 0.88 ACHE (0.43) ACHEGPR119GRIA1KITAOC3
SCHEMBL3879673 0.82 RET (0.40) GPR119GRIA1KITRETCKS1B
SCHEMBL3882036 0.78 GPR119 (0.40) GPR119GRIA1KITRET
SCHEMBL3875573 0.77 DPP4 (0.39) GPR119DPP4
SCHEMBL3874252 0.76 CNR1 (0.42) GPR119GRIA1KITRETPOLB
SCHEMBL3885644 0.76 KIT (0.50) ACHEGPR119KITDDB1CRBN
SCHEMBL3874827 0.73 GPR119 (0.41) GPR119KITPOLB
SCHEMBL25338892 0.73 KIT (0.46) ACHEGPR119GRIA1KITPOLB
SCHEMBL2955911 0.73 POLB (0.45) ACHEGPR119POLBDDB1CRBN
SCHEMBL5275990 0.72 DPP4 (0.64) GPR119DPP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7524847-B2 Fused 1,3-dihydro-imidazole ring compounds EISAI R&D MANAGEMENT CO., LTD. (JP) 2009-04-28 US disclosed
US-7524847-B2 Fused 1,3-dihydro-imidazole ring compounds EISAI R&D MANAGEMENT CO., LTD. (JP) 2009-04-28 US disclosed