SCHEMBL3877928

SCHEMBL3877928

COC(=O)c1cc(F)cc(C(N)C(=O)OC(C)(C)C)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 2/20 0.37
LMNA P02545 2/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
KDM4E B2RXH2 4/20 0.36
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA7 P43166 1/20 0.36
CA9 Q16790 1/20 0.36
CA14 Q9ULX7 1/20 0.36
SLC6A3 Q01959 1/20 0.35
POLB P06746 1/20 0.35
GAA P10253 1/20 0.35
NFKB1 P19838 1/20 0.35
XDH P47989 1/20 0.35
GFER P55789 1/20 0.35
NFKB2 Q00653 1/20 0.35
RELA Q04206 1/20 0.35
FUT7 Q11130 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4180022 1.00 DPP4 (0.37) DPP4LMNAMEN1KMT2AKDM4E
SCHEMBL2569650 0.79 MAPT (0.45) DPP4KDM4ECA12CA1CA2
SCHEMBL12231302 0.75 APP (0.42) DPP4MEN1KMT2AKDM4ECA12
SCHEMBL6629348 0.75 APP (0.42) DPP4MEN1KMT2AKDM4ECA1
SCHEMBL1495951 0.75 DPP4 (0.41) DPP4MEN1KMT2AKDM4ECA12
SCHEMBL23803905 0.75 CA12 (0.46) DPP4LMNAMEN1KMT2AKDM4E
SCHEMBL29738558 0.75 CA12 (0.46) DPP4LMNAMEN1KMT2AKDM4E
SCHEMBL6683190 0.74 CES2 (0.40) DPP4KMT2AKDM4ESLC6A3MAPT
SCHEMBL16952779 0.72 CA12 (0.43) DPP4LMNAMEN1KMT2AKDM4E
SCHEMBL29036907 0.72 SLC6A4 (0.37) SLC6A3FPR2SCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1814846-B1 11BETA-HSD1 INHIBITORS EVOTEC AG (DE) 2009-04-08 EP disclosed
US-20090069323-A1 11beta-hsdi inhibitors EVOTEC AG (DE) 2009-03-12 US disclosed
EP-1814846-A1 11BETA-HSD1 INHIBITORS Evotec AG (DE) 2007-08-08 EP disclosed
WO-2006048330-A1 11ΒΕΤΑ-HSD1 INHIBITORS EVOTEC AG (DE) 2006-05-11 WO disclosed
EP-1655283-A1 11beta-HSD1 Inhibitors Evotec OAI AG (DE) 2006-05-10 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090069323-A1 11beta-hsdi inhibitors HSD3B1, HSD3B2, HSD11B1 DPP4 533/4885LMNA 2473/4885MEN1 1676/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.