SCHEMBL3878084

SCHEMBL3878084

Cc1cccc(-c2ccc(O)cn2)c1

nearest known ligand 0.54

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HSD17B1 P14061 3/20 0.54
HSD17B2 P37059 3/20 0.54
KDM1A O60341 2/20 0.54
IDO1 P14902 1/20 0.49
METAP2 P50579 1/20 0.49
KMO O15229 2/20 0.46
ACHE P22303 2/20 0.45
BCHE P06276 1/20 0.45
XDH P47989 1/20 0.43
CYP3A4 P08684 1/20 0.42
CYP2A6 P11509 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12797772 0.83 CYP3A4 (0.59) HSD17B1HSD17B2KDM1AIDO1METAP2
SCHEMBL12973163 0.83 HSD17B1 (0.59) HSD17B1HSD17B2KDM1AIDO1METAP2
SCHEMBL18573279 0.83 HSD17B1 (0.42) HSD17B1HSD17B2KDM1AACHECYP3A4
SCHEMBL3422110 0.81 IDO1 (0.58) HSD17B1HSD17B2KDM1AIDO1METAP2
SCHEMBL4402515 0.80 HSD17B1 (0.61) HSD17B1HSD17B2KDM1AIDO1METAP2
SCHEMBL23572016 0.79 HSD17B1 (0.69) HSD17B1HSD17B2KDM1AMETAP2ACHE
SCHEMBL14446367 0.79 KDM1A (0.54) HSD17B1HSD17B2KDM1AIDO1METAP2
SCHEMBL14988681 0.79 KDM1A (0.61) HSD17B1HSD17B2KDM1AIDO1METAP2
SCHEMBL30610289 0.79 HSD17B1 (0.69) HSD17B1HSD17B2KDM1AMETAP2ACHE
SCHEMBL15014085 0.79 KDM1A (0.54) HSD17B1HSD17B2KDM1AIDO1METAP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2010485-B1 AZETIDINE DERIVATIVES AS G-PROTEIN COUPLED RECEPTOR (GPR119 ) AGONISTS PROSIDION LTD (GB) 2012-10-17 EP disclosed
US-20090281076-A1 Azetidine Derivatives as G-Protein Coupled Receptor (GPR119) Agonists PROSIDION LIMITED (GB) 2009-11-12 US disclosed
EP-2010485-A1 AZETIDINE DERIVATIVES AS G-PROTEIN COUPLED RECEPTOR (GPR119 ) AGONISTS Prosidion Limited (GB) 2009-01-07 EP disclosed
WO-2007116230-A1 AZETIDINE DERIVATIVES AS G-PROTEIN COUPLED RECEPTOR (GPR119 ) AGONISTS PROSIDION LTD (GB) 2007-10-18 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090281076-A1 Azetidine Derivatives as G-Protein Coupled Receptor (GPR119) Agonists GPR119, GPR39, GIPR HSD17B1 2222/4885HSD17B2 2303/4885KDM1A 2700/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.