SCHEMBL3878656

SCHEMBL3878656

CC(C)C(Nc1nc(-c2ccc(F)c(Cl)c2)cc(N2CCN(c3ncccc3C(F)(F)F)CC2)n1)C(=O)O

nearest known ligand 0.44

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 7/20 0.42
GAA P10253 1/20 0.41
RBP4 P02753 2/20 0.41
TRPA1 O75762 1/20 0.41
TRPV1 Q8NER1 1/20 0.41
NPSR1 Q6W5P4 1/20 0.39
HSD17B10 Q99714 1/20 0.39
GALR2 O43603 1/20 0.39
GALR1 P47211 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3878661 1.00 HSD11B1 (0.42) HSD11B1GAARBP4TRPA1TRPV1
SCHEMBL3880146 0.92 HSD11B1 (0.43) HSD11B1GAARBP4TRPA1TRPV1
SCHEMBL3880138 0.92 HSD11B1 (0.43) HSD11B1GAARBP4TRPA1TRPV1
SCHEMBL3884755 0.89 HSD11B1 (0.45) HSD11B1TRPV1GALR2GALR1
SCHEMBL3882178 0.89 GAA (0.43) HSD11B1GAARBP4TRPA1TRPV1
SCHEMBL3877637 0.85 HSD11B1 (0.46) HSD11B1GAARBP4GALR2GALR1
SCHEMBL3946732 0.82 TRPV1 (0.42) HSD11B1TRPV1
SCHEMBL3880682 0.81 HSD11B1 (0.46) HSD11B1GAARBP4TRPA1TRPV1
SCHEMBL3876842 0.81 HSD11B1 (0.49) HSD11B1TRPV1
SCHEMBL3877152 0.80 HSD11B1 (0.47) HSD11B1GALR2GALR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7566712-B2 Biaryl piperazinyl-pyridine analogues NEUROGEN CORPORATION (US) 2009-07-28 US disclosed
US-7566712-B2 Biaryl piperazinyl-pyridine analogues NEUROGEN CORPORATION (US) 2009-07-28 US disclosed
US-7566712-B2 Biaryl piperazinyl-pyridine analogues NEUROGEN CORPORATION (US) 2009-07-28 US disclosed