SCHEMBL3879174

SCHEMBL3879174

NCCc1ccc(OCC(F)(F)F)cn1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.41
MAPT P10636 2/20 0.41
MAOB P27338 3/20 0.39
HRH1 P35367 1/20 0.38
CACNA1G O43497 1/20 0.36
CACNA1H O95180 1/20 0.36
CNR2 P34972 1/20 0.36
KCNH2 Q12809 1/20 0.36
CACNA1I Q9P0X4 1/20 0.36
GPR3 P46089 1/20 0.35
SCN5A Q14524 1/20 0.35
TAAR1 Q96RJ0 1/20 0.34
CYP2C9 P11712 2/20 0.34
CYP17A1 P05093 1/20 0.34
CYP2C19 P33261 1/20 0.34
CYP1A2 P05177 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
HDAC5 Q9UQL6 1/20 0.34
KDM4E B2RXH2 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL1867868 0.98 MAOB (0.41) ALDH1A1MAPTMAOBHRH1CACNA1G
SCHEMBL507036 0.86 ALDH1A1 (0.43) ALDH1A1MAPTMAOBCACNA1GCACNA1H
SCHEMBL14211870 0.79 CACNA1I (0.40) ALDH1A1MAPTCACNA1GCACNA1HCNR2
SCHEMBL1063185 0.79 CACNA1I (0.40) ALDH1A1MAPTCACNA1GCACNA1HCNR2
SCHEMBL506395 0.79 ALDH1A1 (0.39) ALDH1A1MAPTCACNA1GCACNA1HCNR2
SCHEMBL18172012 0.75 ALDH1A1 (0.50) ALDH1A1MAPTCACNA1GCACNA1HCNR2
SCHEMBL264652 0.75 TAAR1 (0.52) ALDH1A1MAOBHRH1TAAR1KMT2A
SCHEMBL1025383 0.75 TAAR1 (0.52) ALDH1A1MAPTMAOBHRH1TAAR1
SCHEMBL31477886 0.75 TAAR1 (0.52) ALDH1A1MAOBHRH1TAAR1KMT2A
SCHEMBL3889562 0.75 MAOB (0.63) MAOBTAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2010493-A2 PYRIDYL AMIDE T-TYPE CALCIUM CHANNEL ANTAGONISTS Merck & Co., Inc. (US) 2009-01-07 EP disclosed
WO-2007120729-A2 PYRIDYL AMIDE T-TYPE CALCIUM CHANNEL ANTAGONISTS MERCK & CO., INC. (US) 2007-10-25 WO disclosed