SCHEMBL3880561

SCHEMBL3880561

NCCc1ccc(N=C=S)cc1

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RY6 Q15077 1/20 0.76
NOS3 P29474 2/20 0.50
NOS1 P29475 2/20 0.50
NOS2 P35228 2/20 0.50
MIF P14174 1/20 0.46
CA1 P00915 1/20 0.46
CA2 P00918 1/20 0.46
TAAR1 Q96RJ0 8/20 0.45
HTR2A P28223 3/20 0.45
CYP2A6 P11509 2/20 0.45
CYP1A2 P05177 1/20 0.45
KDM4E B2RXH2 1/20 0.45
ALDH1A1 P00352 1/20 0.45
HTR1A P08908 1/20 0.45
ADRA2A P08913 1/20 0.45
SLC6A2 P23975 1/20 0.45
CYP2C19 P33261 1/20 0.45
HTR3A P46098 1/20 0.45
BACE1 P56817 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1853024 0.87 P2RY6 (1.00) P2RY6MIFCA1CA2CYP2A6
SCHEMBL9547715 0.87 P2RY6 (1.00) P2RY6MIFCA1CA2CYP2A6
SCHEMBL16192966 0.83 P2RY6 (0.68) P2RY6NOS3NOS1NOS2MIF
SCHEMBL347652 0.81 P2RY6 (0.79) P2RY6MIFCA1CA2CYP2A6
SCHEMBL6417472 0.79 P2RY6 (0.76) P2RY6MIFCA1CA2CYP2A6
SCHEMBL8503279 0.79 P2RY6 (0.76) P2RY6MIFCA1CA2CYP2A6
SCHEMBL5186242 0.79 P2RY6 (0.76) P2RY6MIFCA1CA2CYP1A2
SCHEMBL27467439 0.79 P2RY6 (0.76) P2RY6MIFCA1CA2CYP2A6
SCHEMBL1193625 0.78 P2RY6 (0.74) P2RY6MIFCA1CA2CYP1A2
SCHEMBL9547731 0.78 P2RY6 (0.74) P2RY6MIFCA1CA2CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240238461-A1 MACROCYCLIC COMPOUNDS AND METHODS OF USE THEREOF JANSSEN BIOTECH, INC. 2024-07-18 US disclosed
EP-1476197-B1 SYNTHESIS OF LIPOPOLYSACCHARIDE-PROTEIN CONJUGATE VACCINES VIA THE LIPID A REGION FOLLOWING REMOVAL OF THE GLYCOSIDIC PHOSPHATE RESIDUE CA NAT RESEARCH COUNCIL (CA) 2009-01-07 EP disclosed
EP-1129092-B1 PORPHYRIN COMPOUNDS, THEIR CONJUGATES AND ASSAY METHODS BASED ON THE USE OF SAID CONJUGATES ARCTIC DIAGNOSTICS OY (FI) 2005-02-23 EP disclosed
US-6740756-B1 POLYAMINO-POLYCARBOXYLIC ACID DERIVATIVES CONTAINING FUSED HETEROCYCLIC KETONE SUBSTITUTED FUNCTIONALITY; LONG LIVED ACTIVITY SMITHKLINE BEECHAM CORPORATION 2004-05-25 US disclosed
US-6582930-B1 Porphyrin for use as diagnostic tools in the food industry and pollution control ARCTIC DIAGNOSTICS OY (FI) 2003-06-24 US disclosed
EP-1095011-A4 NOVEL FLUORESCENT LANTHANIDE CHELATES SMITHKLINE BEECHAM CORP (US) 2003-01-08 EP disclosed
EP-1129092-A1 PORPHYRIN COMPOUNDS, THEIR CONJUGATES AND ASSAY METHODS BASED ON THE USE OF SAID CONJUGATES Arctic Diagnostics OY (FI) 2001-09-05 EP disclosed
EP-1095011-A1 NOVEL FLUORESCENT LANTHANIDE CHELATES SMITHKLINE BEECHAM CORPORATION (US) 2001-05-02 EP disclosed
WO-2000027847-A1 PORPHYRIN COMPOUNDS, THEIR CONJUGATES AND ASSAY METHODS BASED ON THE USE OF SAID CONJUGATES ARCTIC DIAGNOSTICS OY (FI) 2000-05-18 WO disclosed
WO-2000001663-A1 NOVEL FLUORESCENT LANTHANIDE CHELATES SMITHKLINE BEECHAM CORPORATION (US) 2000-01-13 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240238461-A1 MACROCYCLIC COMPOUNDS AND METHODS OF USE THEREOF BDNF, CD47, MAG P2RY6 4603/4885NOS3 1837/4885NOS1 2717/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.