SCHEMBL3883647

SCHEMBL3883647

O=C(O)/C=C/c1cc(-c2ccc(O)cc2)n(C2CCCCC2)n1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 2/20 0.47
ESR1 P03372 5/20 0.41
FABP3 P05413 3/20 0.40
FABP4 P15090 3/20 0.40
S1PR1 P21453 2/20 0.39
RARB P10826 1/20 0.38
CA12 O43570 1/20 0.37
AKR1B10 O60218 1/20 0.37
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
CA3 P07451 1/20 0.37
PKM P14618 1/20 0.37
TYR P14679 1/20 0.37
AKR1B1 P15121 1/20 0.37
CA4 P22748 1/20 0.37
CA6 P23280 1/20 0.37
DPP4 P27487 1/20 0.37
CA5A P35218 1/20 0.37
CA7 P43166 1/20 0.37
CA9 Q16790 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4001179 1.00 PTGS2 (0.47) PTGS2ESR1FABP3FABP4S1PR1
SCHEMBL3866153 0.86 PTGS2 (0.46) PTGS2FABP3FABP4S1PR1RARB
SCHEMBL1131606 0.86 PTGS2 (0.46) PTGS2ESR1FABP3FABP4S1PR1
SCHEMBL1131603 0.83 FABP3 (0.46) PTGS2FABP3FABP4PKM
SCHEMBL1131599 0.83 FABP3 (0.46) PTGS2FABP3FABP4PKM
SCHEMBL12860103 0.82 FABP3 (0.47) PTGS2FABP3FABP4S1PR1RARB
SCHEMBL1131611 0.81 PTGS2 (0.43) PTGS2ESR1FABP3FABP4GCGR
SCHEMBL5861842 0.81 PTGS2 (0.43) PTGS2ESR1FABP3FABP4GCGR
SCHEMBL1131608 0.77 ESR1 (0.40) PTGS2ESR1FABP3FABP4GCGR
SCHEMBL1131325 0.75 CMKLR1 (0.40) PTGS2FABP3FABP4S1PR1CNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1663105-A4 CYCLOALKYL HETEROCYCLES FOR TREATING HEPATITIS C VIRUS BRISTOL MYERS SQUIBB CO (US) 2009-04-15 EP disclosed
US-7112601-B2 Cycloalkyl heterocycles for treating hepatitis C virus BRISTOL-MYERS SQUIBB COMPANY (US) 2006-09-26 US disclosed
EP-1663105-A2 CYCLOALKYL HETEROCYCLES FOR TREATING HEPATITIS C VIRUS Bristol-Myers Squibb Company (US) 2006-06-07 EP disclosed
WO-2005034850-A2 CYCLOALKYL HETEROCYCLES FOR TREATING HEPATITIS C VIRUS BRISTOL-MYERS SQUIBB COMPANY (US) 2005-04-21 WO disclosed
US-20050075376-A1 Cycloalkyl heterocycles for treating Hepatitis C virus BRISTOL-MYERS SQUIBB COMPANY 2005-04-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050075376-A1 Cycloalkyl heterocycles for treating Hepatitis C virus HCCS, NSUN2, HAVCR2 PTGS2 1124/4885ESR1 4488/4885FABP3 3457/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.