SCHEMBL388564

SCHEMBL388564

COC(=O)c1nn(-c2ccccc2)c(=O)cc1O

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.76
SMN1; SMN2 Q16637 4/20 0.68
CYP2C9 P11712 2/20 0.68
CYP2C19 P33261 2/20 0.68
CYP1A2 P05177 1/20 0.68
KMT2A Q03164 3/20 0.68
FHIT P49789 1/20 0.67
MAPK1 P28482 2/20 0.60
RAB9A P51151 2/20 0.57
KDM4E B2RXH2 3/20 0.56
MAPT P10636 4/20 0.53
GAA P10253 3/20 0.53
THRB P10828 1/20 0.53
RECQL P46063 1/20 0.53
L3MBTL1 Q9Y468 1/20 0.53
CYP3A4 P08684 1/20 0.52
NPSR1 Q6W5P4 1/20 0.52
TP53 P04637 2/20 0.51
NPC1 O15118 1/20 0.51
ALOX15 P16050 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11945539 0.86 ALDH1A1 (0.76) ALDH1A1SMN1; SMN2CYP2C9CYP2C19CYP1A2
SCHEMBL25078375 0.86 CYP2C9 (0.68) ALDH1A1SMN1; SMN2CYP2C9CYP2C19CYP1A2
SCHEMBL391859 0.84 KMT2A (0.67) ALDH1A1SMN1; SMN2CYP2C9CYP2C19CYP1A2
SCHEMBL1550557 0.84 ALDH1A1 (0.73) ALDH1A1SMN1; SMN2CYP2C9CYP2C19CYP1A2
SCHEMBL15440699 0.84 KMT2A (0.73) ALDH1A1SMN1; SMN2CYP2C9CYP2C19CYP1A2
SCHEMBL1750835 0.83 KMT2A (0.77) ALDH1A1SMN1; SMN2CYP2C9CYP2C19CYP1A2
SCHEMBL2538523 0.83 ALDH1A1 (0.71) ALDH1A1SMN1; SMN2CYP2C9CYP2C19CYP1A2
SCHEMBL28748456 0.82 ALDH1A1 (0.60) ALDH1A1SMN1; SMN2CYP2C9CYP2C19CYP1A2
SCHEMBL2546655 0.81 ALDH1A1 (0.69) ALDH1A1SMN1; SMN2CYP2C9CYP2C19CYP1A2
SCHEMBL25077819 0.81 ALDH1A1 (0.58) ALDH1A1SMN1; SMN2CYP2C9CYP2C19CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 48 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4667458-A1 PHARMACEUTICAL COMPOSITION FOR TREATMENT OF CANCER, COMPRISING SOS1 INHIBITOR AND ANTICANCER DRUG Kanaph Therapeutics Inc. (KR) 2025-12-24 EP disclosed
WO-2024172631-A1 PHARMACEUTICAL COMPOSITION FOR TREATMENT OF CANCER, COMPRISING SOS1 INHIBITOR AND ANTICANCER DRUG 주식회사 카나프테라퓨틱스 2024-08-22 WO disclosed
CN-118119600-A SOS1 inhibitors and uses thereof 治纳辅医药科技有限公司 2024-05-31 CN disclosed
WO-2023022497-A1 SOS1 INHIBITOR AND USE THEREOF 주식회사 카나프테라퓨틱스 2023-02-23 WO disclosed
WO-2023022497-A1 SOS1 INHIBITOR AND USE THEREOF 주식회사 카나프테라퓨틱스 2023-02-23 WO disclosed
US-10479771-B2 Pyridazinone and pyridone compounds BIOTIE THERAPIES CORPORATION (FI) 2019-11-19 US disclosed
US-20180029995-A1 PYRIDAZINONE AND PYRIDONE COMPOUNDS BIOTIE THERAPIES CORPORATION (FI) 2018-02-01 US disclosed
US-9815795-B2 Pyridazinone and pyridone compounds BIOTIE THERAPIES CORPORATION (FI) 2017-11-14 US disclosed
EP-2683711-B1 NEW PYRIDAZINONE AND PYRIDONE COMPOUNDS BIOTIE THERAPIES CORP (FI) 2017-02-01 EP disclosed
US-20160244414-A1 PYRIDAZINONE AND PYRIDONE COMPOUNDS BIOTIE THERAPIES CORPORATION (FI) 2016-08-25 US disclosed
US-20090143389-A1 HETEROCYCLIC INHIBITORS OF MEK AND METHODS OF USE THEREOF ARRAY BIOPHARMA INC. (US) 2009-06-04 US disclosed
US-20090143579-A1 Heterocyclic Inhibitors of MEK and Methods of Use Thereof ARRAY BIOPHARMA INC. (US) 2009-06-04 US disclosed
US-20090131435-A1 HETEROCYCLIC INHIBITORS OF MEK AND METHODS OF USE ARRAY BIOPHARMA INC. (US) 2009-05-21 US disclosed
US-7517994-B2 Heterocyclic inhibitors of MEK and methods of use thereof ARRAY BIOPHARMA INC. (US) 2009-04-14 US disclosed
EP-2010165-A2 ABNORMAL CANNABIDIOLS AS AGENTS FOR LOWERING INTRAOCULAR PRESSURE Allergan, Inc. (US) 2009-01-07 EP disclosed
WO-2007127711-A2 ABNORMAL CANNABIDIOLS AS AGENTS FOR LOWERING INTRAOCULAR PRESSURE ALLERGAN, INC. (US) 2007-11-08 WO disclosed
US-20070249596-A1 ABNORMAL CANNABIDIOLS AS AGENTS FOR LOWERING INTRAOCULAR PRESSURE ALLERGAN, INC. 2007-10-25 US disclosed
US-20070112038-A1 Heterocyclic inhibitors of MEK and methods of use thereof ARRAY BIOPHARMA INC. 2007-05-17 US disclosed
US-20050256123-A1 Heterocyclic inhibitors of MEK and methods of use thereof ARRAY BIOPHARMA INC. 2005-11-17 US disclosed
US-20050250782-A1 Heterocyclic inhibitors of MEK and methods of use thereof ARRAY BIOPHARMA INC. 2005-11-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (10 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070249596-A1 ABNORMAL CANNABIDIOLS AS AGENTS FOR LOWERING INTRAOCULAR PRESSURE CNR2, CNR1, PTGIR ALDH1A1 3297/4885SMN1; SMN2 4837/4885CYP2C9 539/4885
US-20070112038-A1 Heterocyclic inhibitors of MEK and methods of use thereof NRAS, BRAF, MAPK9 ALDH1A1 1723/4885SMN1; SMN2 3954/4885CYP2C9 144/4885
US-20090131435-A1 HETEROCYCLIC INHIBITORS OF MEK AND METHODS OF USE NRAS, BRAF, MAPK9 ALDH1A1 1962/4885SMN1; SMN2 3942/4885CYP2C9 139/4885
US-20090143389-A1 HETEROCYCLIC INHIBITORS OF MEK AND METHODS OF USE THEREOF NRAS, BRAF, MAPK9 ALDH1A1 1380/4885SMN1; SMN2 3932/4885CYP2C9 178/4885
US-20050250782-A1 Heterocyclic inhibitors of MEK and methods of use thereof NRAS, BRAF, MAPK9 ALDH1A1 1991/4885SMN1; SMN2 4172/4885CYP2C9 130/4885
US-20160244414-A1 PYRIDAZINONE AND PYRIDONE COMPOUNDS XDH, PNPO, PDXK ALDH1A1 259/4885SMN1; SMN2 3199/4885CYP2C9 54/4885
US-20180029995-A1 PYRIDAZINONE AND PYRIDONE COMPOUNDS XDH, PNPO, PDXK ALDH1A1 259/4885SMN1; SMN2 3199/4885CYP2C9 54/4885
US-10479771-B2 Pyridazinone and pyridone compounds XDH, PNPO, PDXK ALDH1A1 259/4885SMN1; SMN2 3199/4885CYP2C9 54/4885
US-20090143579-A1 Heterocyclic Inhibitors of MEK and Methods of Use Thereof NRAS, BRAF, MAPK9 ALDH1A1 2027/4885SMN1; SMN2 4064/4885CYP2C9 134/4885
US-20050256123-A1 Heterocyclic inhibitors of MEK and methods of use thereof NRAS, BRAF, MAPK9 ALDH1A1 1992/4885SMN1; SMN2 4055/4885CYP2C9 136/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.