Iopanoic Acid

Iopanoic Acid

SCHEMBL38976

CCC(Cc1c(I)cc(I)c(N)c1I)C(=O)O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 1.00
CYP2C9 P11712 2/20 1.00
CYP1A2 P05177 2/20 1.00
CHRM1 P11229 1/20 1.00
TBXA2R P21731 1/20 1.00
PDE4A P27815 1/20 1.00
ADRA1A P35348 1/20 1.00
HIF1A Q16665 1/20 1.00
TDP1 Q9NUW8 1/20 0.71
SIRT5 Q9NXA8 1/20 0.38
SLC1A3 P43003 1/20 0.35
SLC1A2 P43004 1/20 0.35
SLC1A1 P43005 1/20 0.35
PPARG P37231 4/20 0.33
CA2 P00918 1/20 0.33
MAPK1 P28482 1/20 0.33
PLA2G10 O15496 1/20 0.32
PLA2G2A P14555 1/20 0.32
NR4A2 P43354 1/20 0.32
EPHX2 P34913 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Iopanoic Acid SCHEMBL29358912 1.00 LMNA (1.00) LMNACYP2C9CYP1A2CHRM1TBXA2R
SCHEMBL18609115 0.88 LMNA (0.79) LMNACYP2C9CYP1A2CHRM1TBXA2R
SCHEMBL8336112 0.88 LMNA (0.78) LMNACYP2C9CYP1A2CHRM1TBXA2R
SCHEMBL18922031 0.88 LMNA (0.78) LMNACYP2C9CYP1A2CHRM1TBXA2R
Iopanoic Acid SCHEMBL31609799 0.85 LMNA (0.74) LMNACYP2C9CYP1A2CHRM1TBXA2R
Iophenoxic Acid SCHEMBL966564 0.83 TDP1 (1.00) LMNACYP2C9CYP1A2CHRM1TBXA2R
SCHEMBL10495750 0.82 CYP1A2 (0.70) LMNACYP2C9CYP1A2CHRM1TBXA2R
SCHEMBL9002219 0.80 LMNA (0.66) LMNACYP2C9CYP1A2CHRM1TBXA2R
SCHEMBL9002211 0.80 LMNA (0.66) LMNACYP2C9CYP1A2CHRM1TBXA2R
SCHEMBL10001207 0.79 LMNA (0.66) LMNACYP2C9CYP1A2CHRM1TBXA2R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 3596 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12582717-B2 Protein based excipient for active pharmaceutical ingredients DISPERSOME IP APS (NL) 2026-03-24 US claimed
US-20260000646-A1 Inhibition of Oral Microbe Biofilms THE UNIVERSITY OF TOLEDO (US) 2026-01-01 US claimed
WO-2025111482-A1 COMPLEXING AGENT SALT FORMULATIONS OF PHARMACEUTICAL COMPOUNDS AT LOW STOICHIOMETRIC RATIOS BEXSON BIOMEDICAL, INC. (US) 2025-05-30 WO claimed
US-20250170279-A1 LIPOSOMAL NANOCARRIER DELIVERY SYSTEM FOR TARGETING ACTIVE CD44 MOLECULE, PREPARATION METHOD THEREFOR, AND USES THEREOF BEIJING INNO MEDICINE CO., LTD. (CN) 2025-05-29 US claimed
US-20250170280-A1 LIPOSOMAL NANOCARRIER DELIVERY SYSTEM FOR TARGETING ACTIVE CD44 MOLECULE, PREPARATION METHOD THEREFOR, AND USES THEREOF BEIJING INNO MEDICINE CO., LTD. (CN) 2025-05-29 US claimed
US-20240293441-A1 NEW THERAPEUTIC USE OF TYPE 2 IODOTHYRONINE DEIODINASE (D2) INHIBITORS CHEIRONTECH S.R.L. (IT) 2024-09-05 US claimed
US-20240226000-A9 TRANSDERMAL PENETRANT FORMULATIONS FOR ADMINISTRATION OF MEDICAMENTS DYVE BIOSCIENCES, INC. 2024-07-11 US claimed
US-20240139003-A1 BIORESORBABLE STENT AND METHOD FOR MANUFACTURING THE SAME INDUSTRY FOUNDATION OF CHONNAM NATIONAL UNIVERSITY (KR) 2024-05-02 US claimed
US-20240130962-A1 TRANSDERMAL PENETRANT FORMULATIONS FOR ADMINISTRATION OF MEDICAMENTS DYVE BIOSCIENCES INC (US) 2024-04-25 US claimed
EP-4346841-A1 NEW THERAPEUTIC USE OF TYPE 2 IODOTHYRONINE DEIODINASE (D2) INHIBITORS Dompé Farmaceutici S.p.A. (IT) 2024-04-10 EP claimed
EP-0649302-A1 THERAPEUTIC AND DIAGNOSTIC USE OF MODIFIED POLYMERIC MICROCAPSULES WALLACE, Sidney (US) 1995-04-26 EP claimed
WO-1995008116-A1 METHOD OF DETECTING CYTOPENIA THAT IS MEDIATED BY DRUG-DEPENDENT ANTIBODY BINDING TO BLOOD CELLS THE BLOOD CENTER OF SOUTHEASTERN WISCONSIN, INC. (US) 1995-03-23 WO claimed
WO-1994027644-A1 IODINATED PARAMAGNETIC CHELATES, AND THEIR USE AS CONTRAST AGENTS BRACCO S.P.A. (IT) 1994-12-08 WO claimed
EP-0414806-B1 HIGH RATIO ACTIVE AGENT:LIPID COMPLEX LIPOSOME CO INC (US) 1994-07-20 EP claimed
WO-1994005335-A1 NEW ORGANIC CONTRAST AGENT ANALOG AND METHOD OF MAKING SAME MOLECULAR BIOSYSTEMS, INC. (US) 1994-03-17 WO claimed
WO-1994002106-A1 THERAPEUTIC AND DIAGNOSTIC USE OF MODIFIED POLYMERIC MICROCAPSULES BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 1994-02-03 WO claimed
EP-0414806-A4 HIGH RATIO ACTIVE AGENT:LIPID COMPLEX 1991-11-13 EP claimed
EP-0414806-A1 HIGH RATIO ACTIVE AGENT:LIPID COMPLEX. LIPOSOME CO INC (US) 1991-03-06 EP claimed
WO-1989011272-A1 HIGH RATIO ACTIVE AGENT:LIPID COMPLEX THE LIPOSOME COMPANY, INC. (US) 1989-11-30 WO claimed
US-4192859-A MEDICAL DIAGNOSIS USING X-RAYS E. R. SQUIBB & SONS, INC. (US) 1980-03-11 US claimed