SCHEMBL3906100

SCHEMBL3906100

O=C1CC(=O)c2cccc(O)c2N1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCNB2 O95067 1/20 0.49
CDK1 P06493 1/20 0.49
CCNB1 P14635 1/20 0.49
GSK3B P49841 1/20 0.49
CCNB3 Q8WWL7 1/20 0.49
RAB9A P51151 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
DRD2 P14416 2/20 0.41
DRD1 P21728 2/20 0.41
DRD4 P21917 2/20 0.41
DRD5 P21918 2/20 0.41
DRD3 P35462 2/20 0.41
AHR P35869 1/20 0.41
MAOA P21397 2/20 0.39
TDP2 O95551 4/20 0.39
CASP7 P55210 2/20 0.39
CASP3 P42574 1/20 0.39
CASP9 P55211 1/20 0.39
CASP6 P55212 1/20 0.39
CASP8 Q14790 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13312397 0.78 GSK3B (0.41) CCNB2CDK1CCNB1GSK3BCCNB3
SCHEMBL8765618 0.78 SRD5A1 (0.41) AHRTDP2CASP7CASP3CASP9
SCHEMBL4411843 0.77 AHR (0.61) CCNB2CDK1CCNB1GSK3BCCNB3
SCHEMBL13312445 0.76 BRD4 (0.44) GSK3BAHRTDP2CASP7CASP3
SCHEMBL5688415 0.73 GSK3B (0.74) CCNB2CDK1CCNB1GSK3BCCNB3
SCHEMBL30319806 0.73 GSK3B (0.74) CCNB2CDK1CCNB1GSK3BCCNB3
SCHEMBL5332282 0.71 CES1 (0.60) GSK3BMAOACASP7CASP3CASP6
SCHEMBL31244367 0.71 CES1 (0.60) GSK3BMAOACASP7CASP3CASP6
SCHEMBL1050699 0.68 AHR (0.57) CCNB2CDK1CCNB1GSK3BCCNB3
SCHEMBL13439628 0.68 MAOA (0.56) MAOACASP7ALDH1A1MAPTALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1954689-A4 N-SUBSTITUTED-1H-QUINOLINE-2, 4-DIONES, PREPARATION METHOD THEREOF, AND PHARMACEUTICAL COMPOSITION CONTAINING THE SAME KOREA RES INST CHEM TECH (KR) 2009-09-02 EP claimed
EP-1954689-A1 N-SUBSTITUTED-1H-QUINOLINE-2, 4-DIONES, PREPARATION METHOD THEREOF, AND PHARMACEUTICAL COMPOSITION CONTAINING THE SAME KOREA RESEARCH INSTITUTE OF CHEMICAL TECHNOLOGY (KR) 2008-08-13 EP claimed
WO-2007032572-A1 N-SUBSTITUTED-1H-QUINOLINE-2, 4-DIONES, PREPARATION METHOD THEREOF, AND PHARMACEUTICAL COMPOSITION CONTAINING THE SAME KOREA RESERACH INSTITUTE OF CHEMICAL TECHNOLOGY (KR) 2007-03-22 WO claimed
EP-1650190-A1 3-aryl-3-methyl-quinoline-2,4-diones, preparation method thereof and pharmaceutical composition containing same Korea Research Institute of Chemical Technology (KR) 2006-04-26 EP disclosed