SCHEMBL39114

SCHEMBL39114

C(=CCN(c1ccccc1)c1ccccc1)CN(c1ccccc1)c1ccccc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.38
MAOB P27338 1/20 0.38
KDM4E B2RXH2 4/20 0.36
MTNR1A P48039 1/20 0.36
MTNR1B P49286 1/20 0.36
TAAR1 Q96RJ0 1/20 0.36
ALDH1A1 P00352 3/20 0.35
NPSR1 Q6W5P4 1/20 0.35
ALOX15 P16050 1/20 0.35
ESR1 P03372 1/20 0.34
L3MBTL1 Q9Y468 2/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
MAPT P10636 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
S1PR1 P21453 1/20 0.33
TSHR P16473 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9016977 1.00 KCNH2 (0.38) KCNH2MAOBKDM4EMTNR1AMTNR1B
SCHEMBL9429468 0.84 MEN1 (0.49) KCNH2MAOBKDM4EL3MBTL1CYP1A2
SCHEMBL9016966 0.83 TK1 (0.43) KCNH2MAOBALDH1A1CYP2C19TSHR
SCHEMBL9016968 0.83 TK1 (0.43) KCNH2MAOBALDH1A1CYP2C19TSHR
SCHEMBL39946 0.81 ESR1 (0.44) KCNH2KDM4EALDH1A1ESR1CYP1A2
SCHEMBL9818045 0.81 ESR1 (0.44) KCNH2KDM4EALDH1A1ESR1CYP1A2
SCHEMBL5077351 0.80 KDM4E (0.37) KCNH2KDM4EMTNR1AMTNR1BNPSR1
SCHEMBL2227806 0.80 MAPT (0.38) KCNH2KDM4EMTNR1AMTNR1BTAAR1
SCHEMBL5077354 0.80 KDM4E (0.37) KCNH2KDM4EMTNR1AMTNR1BNPSR1
SCHEMBL3293008 0.79 KCNH2 (0.35) KCNH2KDM4EMTNR1AMTNR1BTAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 2602 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240182674-A1 USE OF A STABILIZER COMPOSITION FOR STABILIZING HALOGEN-FREE RECYCLED THERMOPLASTICS, STABILIZER COMPOSITION, MASTER BATCH OR CONCENTRATE, STABILIZED PLASTIC COMPOSITION, PROCESS FOR STABILIZING HALOGEN-FREE RECYCLED THERMOPLASTICS, AND USE OF COMPOSITIONS Fraunhofer-Gesellschaft zur Förderung der angewandten Forschung e.V. (DE) 2024-06-06 US claimed
EP-4308638-A1 USE OF A STABILIZER COMPOSITION FOR STABILIZING POLYOLEFIN RECYCLATES, STABILIZER COMPOSITION, MASTER BATCH CONCENTRATE, PLASTIC COMPOSITION, MOLDING COMPOUND OR MOLDING, METHOD FOR STABILIZING A POLYOLEFIN RECYCLATE AND USE OF A PLASTIC COMPOSITION Fraunhofer-Gesellschaft zur Förderung der angewandten Forschung e.V. (DE) 2024-01-24 EP claimed
EP-4301809-A1 USE OF A STABILIZER COMPOSITION FOR STABILIZING HALOGEN-FREE RECYCLED THERMOPLASTICS, STABILIZER COMPOSITION, MASTER BATCH OR CONCENTRATE, STABILIZED PLASTIC COMPOSITION, PROCESS FOR STABILIZING HALOGEN-FREE RECYCLED THERMOPLASTICS, AND USE OF COMPOSITIONS Fraunhofer-Gesellschaft zur Förderung der angewandten Forschung e.V. (DE) 2024-01-10 EP claimed
WO-2022194672-A1 USE OF A STABILIZER COMPOSITION FOR STABILIZING POLYOLEFIN RECYCLATES, STABILIZER COMPOSITION, MASTER BATCH CONCENTRATE, PLASTIC COMPOSITION, MOLDING COMPOUND OR MOLDING, METHOD FOR STABILIZING A POLYOLEFIN RECYCLATE AND USE OF A PLASTIC COMPOSITION Fraunhofer-Gesellschaft zur Förderung der angewandten Forschung e.V. (DE) 2022-09-22 WO claimed
WO-2022184596-A1 USE OF A STABILIZER COMPOSITION FOR STABILIZING HALOGEN-FREE RECYCLED THERMOPLASTICS, STABILIZER COMPOSITION, MASTER BATCH OR CONCENTRATE, STABILIZED PLASTIC COMPOSITION, PROCESS FOR STABILIZING HALOGEN-FREE RECYCLED THERMOPLASTICS, AND USE OF COMPOSITIONS Fraunhofer-Gesellschaft zur Förderung der angewandten Forschung e.V. (DE) 2022-09-09 WO claimed
EP-2920236-B1 POLYMER COMPOSITION HAVING IMPROVED LONG-TERM STABILITY, MOULDED PARTS PRODUCED THEREFROM AND INTENDED USES THEREOF FRAUNHOFER GES FORSCHUNG (DE) 2019-06-05 EP claimed
US-10233298-B2 Polyurethane foams based on polyether carbonate polyols COVESTRO DEUTSCHLAND AG (DE) 2019-03-19 US claimed
EP-3250620-B1 POLYURETHANE FOAMS BASED ON POLYETHER CARBONATE POLYOLS COVESTRO DEUTSCHLAND AG (DE) 2018-11-14 EP claimed
US-20180265623-A1 POLYURETHANE FOAMS BASED ON POLYETHER CARBONATE POLYOLS COVESTRO DEUTSCHLAND AG (DE) 2018-09-20 US claimed
EP-3134449-A1 POLYURETHANE FOAMS BASED ON POLYETHER CARBONATE POLYOLS Covestro Deutschland AG (DE) 2017-03-01 EP claimed
US-20170044341-A1 POLYURETHANE FOAMS BASED ON POLYETHER CARBONATE POLYOLS COVESTRO DEUTSCHLAND AG (DE) 2017-02-16 US claimed
US-20160272789-A1 POLYMER COMPOSITION WITH IMPROVED LONG-TERM STABILITY, MOULDED PARTS PRODUCED HEREFROM AND ALSO PURPOSES OF USE FRAUNHOFER-GESELLACHAFT ZUR FÖRDERUNG DER ANGEWANDTEN FORSCHUNG E.V. (DE) 2016-09-22 US claimed
US-9181481-B2 Liquid crystal display device and method of manufacturing the same SAMSUNG DISPLAY CO., LTD. (KR) 2015-11-10 US claimed
WO-2015162125-A1 POLYURETHANE FOAMS BASED ON POLYETHER CARBONATE POLYOLS BAYER MATERIAL SCIENCE AG (DE) 2015-10-29 WO claimed
EP-0514333-A2 Substituted 1,4-diamino-2-butene stabilizers and stabilized compositions CIBA-GEIGY AG (CH) 1992-11-19 EP claimed
JP-3093751-A None JP disclosed
EP-4731727-A1 HALF-WAVE PLATE Merck Patent GmbH (DE) 2026-04-29 EP disclosed
EP-0454622-A1 Alkenyl substituted stabilizers CIBA-GEIGY AG (CH) 1991-10-30 EP disclosed
JP-H0393751-A STABILISER FOR BUTENYL AROMATIC AMINE CIBA GEIGY AG 1991-04-18 JP disclosed
EP-0417036-A2 Butenyl aromatic amine stabilizers CIBA-GEIGY AG (CH) 1991-03-13 EP disclosed