SCHEMBL3915355

SCHEMBL3915355

FC(F)(F)c1ccc(CSc2nnc(-c3ccco3)n2-c2ccccc2)cc1

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 11/20 0.76
KMT2A Q03164 3/20 0.76
KDM4E B2RXH2 3/20 0.76
MEN1 O00255 2/20 0.76
LMNA P02545 2/20 0.76
PKM P14618 1/20 0.57
RAB9A P51151 3/20 0.57
SMN1; SMN2 Q16637 2/20 0.57
GAA P10253 1/20 0.57
TSHR P16473 10/20 0.56
POLB P06746 4/20 0.56
USP2 O75604 2/20 0.56
NPC1 O15118 2/20 0.56
HPGD P15428 3/20 0.54
NPSR1 Q6W5P4 2/20 0.54
HTT P42858 1/20 0.54
OPRK1 P41145 1/20 0.53
MITF O75030 1/20 0.53
MAPT P10636 1/20 0.53
ATM Q13315 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11511155 0.85 ALDH1A1 (0.69) ALDH1A1KMT2AKDM4EMEN1LMNA
SCHEMBL14133313 0.79 ALDH1A1 (0.67) ALDH1A1KMT2AKDM4EMEN1LMNA
SCHEMBL13831408 0.78 POLB (0.65) ALDH1A1KMT2AKDM4EMEN1GAA
SCHEMBL11510495 0.78 ALDH1A1 (0.73) ALDH1A1KMT2AKDM4EMEN1LMNA
SCHEMBL18997268 0.77 ALDH1A1 (0.64) ALDH1A1KMT2AKDM4EMEN1LMNA
SCHEMBL3905153 0.76 TSHR (0.64) ALDH1A1KMT2AMEN1LMNAPKM
SCHEMBL13401419 0.75 POLB (0.77) ALDH1A1KMT2AKDM4EMEN1LMNA
SCHEMBL6404149 0.75 ALDH1A1 (0.64) ALDH1A1KMT2AKDM4EMEN1LMNA
SCHEMBL3904525 0.72 ALDH1A1 (1.00) ALDH1A1KMT2AKDM4EMEN1LMNA
SCHEMBL31160371 0.71 LMNA (0.53) ALDH1A1KMT2AMEN1LMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7563905-B2 Triazole derivatives and method of using the same to treat HIV infections WYETH (US) 2009-07-21 US claimed
WO-2005090320-A2 TRIAZOLE DERIVATIVES AND METHOD OF USING THE SAME TO TREAT HIV INFECTIONS WYETH (US) 2005-09-29 WO claimed
US-20050209287-A1 Triazole derivatives and method of using the same to treat HIV infections WYETH 2005-09-22 US claimed
US-7563905-B2 Triazole derivatives and method of using the same to treat HIV infections WYETH (US) 2009-07-21 US disclosed
WO-2005090320-A2 TRIAZOLE DERIVATIVES AND METHOD OF USING THE SAME TO TREAT HIV INFECTIONS WYETH (US) 2005-09-29 WO disclosed
US-20050209287-A1 Triazole derivatives and method of using the same to treat HIV infections WYETH 2005-09-22 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050209287-A1 Triazole derivatives and method of using the same to treat HIV infections CYP3A43, XDH, AKR1C3 ALDH1A1 430/4885KMT2A 2209/4885KDM4E 2734/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.