SCHEMBL3915728

SCHEMBL3915728

Cn1c(Oc2ccccc2)ncc(-c2ccc(O)c(F)c2)c1=O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MET P08581 8/20 0.42
HGF P14210 1/20 0.42
MST1R Q04912 1/20 0.42
ALDH1A1 P00352 5/20 0.41
CYP1A2 P05177 5/20 0.41
CYP3A4 P08684 5/20 0.41
HSD17B10 Q99714 5/20 0.41
HPGD P15428 2/20 0.41
TSHR P16473 2/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
COMT P21964 2/20 0.41
USP2 O75604 3/20 0.41
CYP2C9 P11712 3/20 0.41
CASP1 P29466 2/20 0.41
CASP7 P55210 2/20 0.41
MIF P14174 1/20 0.39
FEN1 P39748 3/20 0.39
ACMSD Q8TDX5 1/20 0.37
HIF1A Q16665 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3912098 0.82 MET (0.51) METHGFMST1RFEN1
SCHEMBL2379712 0.77 MET (0.58) METHGFMST1RCYP3A4MIF
SCHEMBL2288757 0.77 MET (0.58) METHGFMST1RALDH1A1CYP1A2
SCHEMBL3912607 0.76 MIF (0.37) METHGFMST1RHSD17B10COMT
SCHEMBL2861659 0.75 ALDH1A1 (0.39) ALDH1A1CYP1A2CYP3A4HSD17B10HPGD
SCHEMBL2280129 0.75 GAA (0.53) METHGFMST1RALDH1A1CYP1A2
SCHEMBL2855704 0.70 MET (0.58) METHGFMST1RCYP1A2USP2
SCHEMBL3117756 0.70 KDM1A (0.40) METCOMTMIFFEN1
SCHEMBL3912756 0.69 HTT (0.47) ALDH1A1CYP1A2CYP3A4HSD17B10HPGD
SCHEMBL3985621 0.68 MEN1 (0.41) METCYP1A2HSD17B10MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110053931-A1 QUINOLINE COMPOUNDS AND METHODS OF USE GAUDINO JOHN 2011-03-03 US disclosed
EP-2032538-A2 QUINOLINE COMPOUNDS AND METHODS OF USE Array Biopharma, Inc. (US) 2009-03-11 EP disclosed
WO-2007146824-A2 QUINOLINE COMPOUNDS AND METHODS OF USE ARRAY BIOPHARMA INC. (US) 2007-12-21 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110053931-A1 QUINOLINE COMPOUNDS AND METHODS OF USE TK1, ABL1, ROR1 MET 563/4885HGF 1991/4885MST1R 413/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.