Dansylsarcosine

Dansylsarcosine

SCHEMBL39162

CN(C)c1cccc2c(S(=O)(=O)N(C)CC(=O)O)cccc12

nearest known ligand 0.61

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Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 2/20 0.61
CYP1A2 P05177 1/20 0.61
CYP2C19 P33261 1/20 0.61
HTT P42858 1/20 0.61
HIF1A Q16665 1/20 0.61
TDP1 Q9NUW8 1/20 0.61
CA2 P00918 1/20 0.55
KEAP1 Q14145 2/20 0.52
NFE2L2 Q16236 2/20 0.52
F2 P00734 3/20 0.51
PRSS1 P07477 3/20 0.51
PRSS2 P07478 3/20 0.51
PRSS3 P35030 3/20 0.51
EDNRA P25101 1/20 0.49
HDAC6 Q9UBN7 3/20 0.48
HDAC3 O15379 2/20 0.48
HDAC1 Q13547 2/20 0.48
HDAC2 Q92769 2/20 0.48
NCOR2 Q9Y618 2/20 0.48
KMT2A Q03164 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Dansylsarcosine SCHEMBL30586115 1.00 L3MBTL1 (0.61) L3MBTL1CYP1A2CYP2C19HTTHIF1A
Dansylsarcosine SCHEMBL23850005 0.89 CYP1A2 (0.50) L3MBTL1CYP1A2CYP2C19HTTHIF1A
Dansylsarcosine SCHEMBL30745135 0.89 CYP1A2 (0.50) L3MBTL1CYP1A2CYP2C19HTTHIF1A
SCHEMBL15627403 0.84 CYP1A2 (0.56) L3MBTL1CYP1A2CYP2C19HTTHIF1A
Dansylsarcosine SCHEMBL5500548 0.84 L3MBTL1 (0.45) L3MBTL1CYP1A2CYP2C19HTTHIF1A
SCHEMBL11888757 0.82 KEAP1 (0.66) L3MBTL1CA2KEAP1NFE2L2PRSS1
SCHEMBL26005791 0.82 CYP1A2 (0.77) L3MBTL1CYP1A2CYP2C19HTTHIF1A
SCHEMBL12964231 0.81 CYP1A2 (0.62) L3MBTL1CYP1A2CYP2C19HTTHIF1A
SCHEMBL14178940 0.81 CYP1A2 (0.59) L3MBTL1CYP1A2CYP2C19HTTHIF1A
SCHEMBL39163 0.80 ALDH1A1 (0.48) L3MBTL1KEAP1NFE2L2ALDH1A1MCL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 3748 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3612842-B1 METHODS FOR DETERMINING THE RELATIVE BINDING CAPACITY OF ALBUMIN FRAUNHOFER GES FORSCHUNG (DE) 2025-11-26 EP claimed
CN-119993473-A System and method for predicting long-term prognosis of liver disease patient 上海交通大学医学院附属瑞金医院 2025-05-13 CN claimed
EP-3884280-B1 METHODS AND KITS FOR DETECTING LIVER DYSFUNCTION IN A SUBJECT INST NAT SANTE RECH MED (FR) 2024-01-17 EP claimed
US-20220018852-A1 METHODS AND KITS FOR DETECTING LIVER DYSFUNCTION IN A SUBJECT CENTRE HOSPITALIER REGIONAL UNIVERSITAIRE DE LIMOGES (FR) 2022-01-20 US claimed
EP-3884280-A1 METHODS AND KITS FOR DETECTING LIVER DYSFUNCTION IN A SUBJECT Institut National de la Santé et de la Recherche Médicale (INSERM) (FR) 2021-09-29 EP claimed
CN-101175766-B Albumin solution ALBUTEC GMBH 2015-04-29 CN claimed
US-8476081-B2 Assay for evaluating affinity and specificity of ligand-albumin binding JANSSEN PHARMACEUTICA NV (BE) 2013-07-02 US claimed
US-20110124120-A1 ASSAY FOR EVALUATING AFFINITY AND SPECIFICITY OF LIGAND-ALBUMIN BINDING JANSSEN PHARMACEUTICA N.V. (BE) 2011-05-26 US claimed
US-20100240602-A1 METHODS AND COMPOSITIONS FOR OPTIMIZING BLOOD AND TISSUE STABILITY OF CAMPTOTHECIN AND OTHER ALBUMIN-BINDING THERAPEUTIC COMPOUNDS BURKE THOMAS G 2010-09-23 US claimed
EP-1315973-B1 INDIRECT METHOD FOR THE QUANTITATIVE ANALYSIS OF THE BINDING CAPACITY PRESENT IN AN AQUEOUS PROTEIN SOLUTION GAMBRO LUNDIA AB (SE) 2009-07-29 EP claimed
JP-2003501487-A 2003-01-14 JP claimed
JP-2002544523-A 2002-12-24 JP claimed
US-20020193318-A1 Methods and compositions for optimizing blood and tissue stability of camptothecin and other albumin-binding therapeutic compounds NEW CENTURY PHARMACEUTICALS, INC. 2002-12-19 US claimed
WO-2002074246-A2 METHOD AND COMPOSITIONS FOR OPTIMIZING BLOOD AND TISSUE STABILITY OF CAMPTOTHECIN AND OTHER ALBUMIN-BINDING THERAPEUTIC COMPOUNDS NEW CENTURY PHARMACEUTICALS, INC. (US) 2002-09-26 WO claimed
EP-1185305-A1 LIGAND-CONJUGATED OLIGOMERIC COMPOUNDS ISIS PHARMACEUTICALS, INC. (US) 2002-03-13 EP claimed
EP-1180244-A2 HIGH TROUGHPUT ASSAY SYSTEMS AND METHODS Caliper Technologies Corporation (US) 2002-02-20 EP claimed
WO-2000076554-A1 LIGAND-CONJUGATED OLIGOMERIC COMPOUNDS ISIS PHARMACEUTICALS, INC. (US) 2000-12-21 WO claimed
WO-2000070353-A2 HIGH THROUGHPUT ASSAY SYSTEMS AND METHODS CALIPER TECHNOLOGIES CORP. (US) 2000-11-23 WO claimed
US-5541633-A Ink jet printing of concealed images on carbonless paper XEROX CORPORATION (US) 1996-07-30 US claimed
US-5286286-A Containing diethylene glycol monobutyl ether, glycerol, and a dansyl or porphyrin chromophores XEROX CORPORATION (US) 1994-02-15 US claimed